All Products

Featured Products

Newest Products

Research Areas

PERK Products

or product name starting with: A   B   C   D   E   F   G   H   I   J   K   L   M   N   O   P   Q   R   S   T   U   V   W   X   Y   Z  
406190
TG101209
featured
TG101209 is a novel and potent JAK2 inhibitor, which induced dose- and time-dependent cytotoxicity i…
401470
GDC-0879
featured
GDC-0879 is a highly selective, potent, and orally bioavailable RAF small-molecule inhibitor. In GDC…
406200
G-573
featured
G-573 is an allosteric inhibitor of MEK that is both potent and selective. The IC(50) value for pERK…
200771
CI-1040
featured
CI-1040, also known as PD184352, is a MEK inhibitor, which demonstrated in vivo activity in preclini…
205903
RXDX-105 (CEP-32496)
featured
RXDX-105, also known as Agerafenib, CEP-32496 and AC013773, is an orally available v-raf murine sarc…
406197
SL327
featured
SL327 is a MEK inhibitor. SL327 blocks acquisition but not expression of lithium-induced conditioned…
206139
Gilteritinib
featured
Gilteritinib, also known as ASP2215, is a potent FLT3/AXL inhibitor, which showed potent antileukemi…
406230
GSK2656157
featured
GSK2656157 is an ATP-competitive inhibitor of PERK enzyme activity with an IC50 of 0.9 nM. It is hig…
406393
GSK2606414
featured
GSK2606414 is an orally available, potent, and selective PERK inhibitor. GSK2606414 inhibits PERK ac…