EP6
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MedKoo CAT#: 558412

CAS#: 1353567-32-4

Description: EP6 is a 5-lipoxygenase (5-LO) inhibitor. 5-LO is a crucial enzyme of the arachidonic acid (AA) cascade and catalyzes the formation of bioactive leukotrienes (LTs) which are involved in inflammatory diseases and allergic reactions.

Chemical Structure

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EP6
CAS# 1353567-32-4
Instruction

Theoretical Analysis

MedKoo Cat#: 558412
Name: EP6
CAS#: 1353567-32-4
Chemical Formula: C24H30N4O
Exact Mass: 390.24
Molecular Weight: 390.530
Elemental Analysis: C, 73.81; H, 7.74; N, 14.35; O, 4.10

Price and Availability

Size Price Availability Quantity
50mg USD 450 2 Weeks
100mg USD 750 2 Weeks
200mg USD 1250 2 Weeks
500mg USD 2650 2 Weeks
1g USD 3850 2 Weeks
2g USD 5850 2 Weeks
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Related CAS #: 1353567-32-4    

Synonym: EP6; EP-6; EP 6;

IUPAC/Chemical Name: N-Cyclohexyl-6-methyl-2-[4-(4-morpholinyl)phenyl]-imidazo[1,2-a]pyridin-3-amine

InChi Key: ITCJJNJMYCQGTM-UHFFFAOYSA-N

InChi Code: InChI=1S/C24H30N4O/c1-18-7-12-22-26-23(24(28(22)17-18)25-20-5-3-2-4-6-20)19-8-10-21(11-9-19)27-13-15-29-16-14-27/h7-12,17,20,25H,2-6,13-16H2,1H3

SMILES Code: CC1=CN2C(C=C1)=NC(C3=CC=C(N4CCOCC4)C=C3)=C2NC5CCCCC5

Appearance: Solid powder

Purity: >98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility: Soluble in DMSO

Shelf Life: >3 years if stored properly

Drug Formulation: This drug may be formulated in DMSO

Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code: 2934.99.03.00

More Info:

Biological target:
In vitro activity:
In vivo activity:

Preparing Stock Solutions

The following data is based on the product molecular weight 390.53 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
Formulation protocol:
In vitro protocol:
In vivo protocol:

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