Tameridone

    WARNING: This product is for research use only, not for human or veterinary use.

MedKoo CAT#: 585092

CAS#: 102144-78-5

Description: Tameridone is a sedative used for cattle.

Chemical Structure

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Tameridone
CAS# 102144-78-5
Instruction

Theoretical Analysis

MedKoo Cat#: 585092
Name: Tameridone
CAS#: 102144-78-5
Chemical Formula: C22H26N6O2
Exact Mass: 406.21
Molecular Weight: 406.490
Elemental Analysis: C, 65.01; H, 6.45; N, 20.68; O, 7.87

Price and Availability

This product is not in stock, which may be available by custom synthesis. For cost-effective reason, minimum order is 1g (price is usually high, lead time is 2~3 months, depending on the technical challenge). Quote less than 1g will not be provided. To request quote, please email to sales @medkoo.com or click below button.
Note: Price will be listed if it is available in the future.

Request quote for custom synthesis

Synonym: Tameridone; R 51163; R 51 163

IUPAC/Chemical Name: 1H-Purine-2,6-dione, 3,7-dihydro-7-(2-(4-(1H-indol-3-yl)-1-piperidinyl)ethyl)-1,3-dimethyl-

InChi Key: OJOSYHJYEWUYGU-UHFFFAOYSA-N

InChi Code: InChI=1S/C22H26N6O2/c1-25-20-19(21(29)26(2)22(25)30)28(14-24-20)12-11-27-9-7-15(8-10-27)17-13-23-18-6-4-3-5-16(17)18/h3-6,13-15,23H,7-12H2,1-2H3

SMILES Code: O=C(N1C)N(C)C2=C(N(CCN3CCC(C4=CNC5=C4C=CC=C5)CC3)C=N2)C1=O

Appearance: Solid powder

Purity: >98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility: Soluble in DMSO

Shelf Life: >3 years if stored properly

Drug Formulation: This drug may be formulated in DMSO

Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code: 2934.99.9001

More Info:

Biological target:
In vitro activity:
In vivo activity:

Preparing Stock Solutions

The following data is based on the product molecular weight 406.49 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
Formulation protocol:
In vitro protocol:
In vivo protocol:

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1: Haigh JC, Gates CC. Capture of wood bison (Bison bison athabascae) using carfentanil-based mixtures. J Wildl Dis. 1995 Jan;31(1):37-42. PubMed PMID: 7563422.

2: Renecker LA, Bertwistle J, Kozak HM, Hudson RJ, Chabot D, MacLean S. R51163 as a sedative for handling and transporting plains bison and wapiti. J Wildl Dis. 1992 Apr;28(2):236-41. PubMed PMID: 1602574.

3: Schwartz CC, Hundertmark KJ, Lance WR. Effects of R51163 on intake and metabolism in moose. J Wildl Dis. 1991 Jan;27(1):119-22. PubMed PMID: 2023310.

4: Jiang YQ, Zuo CX. [Studies of chemical constituents from Tamarix chinensis Lour]. Yao Xue Xue Bao. 1988;23(10):749-55. Chinese. PubMed PMID: 3257027.

5: Degryse AD, Ooms LA. Clinical evaluation of R 51163, a new sedative in cattle. J Vet Pharmacol Ther. 1986 Dec;9(4):376-84. PubMed PMID: 3806779.