Cafaminol

    WARNING: This product is for research use only, not for human or veterinary use.

MedKoo CAT#: 461302

CAS#: 30924-31-3

Description: Cafaminol also known as methylcoffanolamine, is a vasoconstrictor and anticatarrhal of the methylxanthine family related to caffeine which is used as a nasal decongestant

Chemical Structure

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Cafaminol
CAS# 30924-31-3
Instruction

Theoretical Analysis

MedKoo Cat#: 461302
Name: Cafaminol
CAS#: 30924-31-3
Chemical Formula: C11H17N5O3
Exact Mass: 267.13
Molecular Weight: 267.280
Elemental Analysis: C, 49.43; H, 6.41; N, 26.20; O, 17.96

Price and Availability

This product is not in stock, which may be available by custom synthesis. For cost-effective reason, minimum order is 1g (price is usually high, lead time is 2~3 months, depending on the technical challenge). Quote less than 1g will not be provided. To request quote, please email to sales @medkoo.com or click below button.
Note: Price will be listed if it is available in the future.

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Synonym: Cafaminol; Cafaminolum; G 1; G-1; G1; Methylcoffanolamine; Rhinetten; Rhinoptil;

IUPAC/Chemical Name: 8-((2-hydroxyethyl)(methyl)amino)-1,3,7-trimethyl-3,7-dihydro-1H-purine-2,6-dione

InChi Key: ZGNRRVAPHPANFI-UHFFFAOYSA-N

InChi Code: InChI=1S/C11H17N5O3/c1-13(5-6-17)10-12-8-7(14(10)2)9(18)16(4)11(19)15(8)3/h17H,5-6H2,1-4H3

SMILES Code: O=C(N(C1=O)C)N(C2=C1N(C(N(CCO)C)=N2)C)C

Appearance: Solid powder

Purity: >98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility: Soluble in DMSO

Shelf Life: >3 years if stored properly

Drug Formulation: This drug may be formulated in DMSO

Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code: 2934.99.03.00

More Info:

Biological target:
In vitro activity:
In vivo activity:

Preparing Stock Solutions

The following data is based on the product molecular weight 267.28 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
Formulation protocol:
In vitro protocol:
In vivo protocol:

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1: Rogowski M, Chodynicki S. [Use of the preparation Cafaminol in the treatment of acute rhinitis]. Wiad Lek. 1985 Oct 15;38(20):1437-40. Polish. PubMed PMID: 3913153.

2: Walther H, Köhler E. [Human pharmacologic studies on the biologic availability and resorption of cafaminol (AWD) (proceedings)]. Pharmazie. 1979 May-Jun;34(5-6):375-6. German. PubMed PMID: 515164.