TMCB
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    WARNING: This product is for research use only, not for human or veterinary use.

MedKoo CAT#: 562418

CAS#: 905105-89-7

Description: TMCB is a dual-kinase inhibitor. It acts by inhibiting both casein kinase 2 (CK2) and extracellular-signal-regulated kinase 8 (ERK8).

Chemical Structure

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TMCB
CAS# 905105-89-7
Instruction

Theoretical Analysis

MedKoo Cat#: 562418
Name: TMCB
CAS#: 905105-89-7
Chemical Formula: C11H9Br4N3O2
Exact Mass: 530.74
Molecular Weight: 534.820
Elemental Analysis: C, 24.70; H, 1.70; Br, 59.76; N, 7.86; O, 5.98

Price and Availability

Size Price Availability Quantity
10mg USD 270
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Synonym: TMCB;

IUPAC/Chemical Name: 2-(4,5,6,7-Tetrabromo-2-(dimethylamino)-1H-benzo[d]imidazol-1-yl)acetic acid

InChi Key: PHAOTASRLQMKBE-UHFFFAOYSA-N

InChi Code: InChI=1S/C11H9Br4N3O2/c1-17(2)11-16-9-7(14)5(12)6(13)8(15)10(9)18(11)3-4(19)20/h3H2,1-2H3,(H,19,20)

SMILES Code: O=C(O)CN1C(N(C)C)=NC2=C(Br)C(Br)=C(Br)C(Br)=C12

Appearance: Solid powder

Purity: >98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility: Soluble in DMSO

Shelf Life: >2 years if stored properly

Drug Formulation: This drug may be formulated in DMSO

Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code: 2934.99.9001

More Info:

Biological target:
In vitro activity:
In vivo activity:

Preparing Stock Solutions

The following data is based on the product molecular weight 534.82 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
Formulation protocol:
In vitro protocol:
In vivo protocol:

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