WARNING: This product is for research use only, not for human or veterinary use.
MedKoo CAT#: 318407
CAS#: 125-53-1 (free base)
Description: Oxyphencyclimine is a muscarinic receptor antagonist (MRA) anticholinergic drug (trade name Daricon) used in treating peptic ulcers.
MedKoo Cat#: 318407
CAS#: 125-53-1 (free base)
Chemical Formula: C20H28N2O3
Exact Mass: 344.20999
Molecular Weight: 344.46
Elemental Analysis: C, 69.74; H, 8.19; N, 8.13; O, 13.93
This product is not in stock, which may be available by custom synthesis.
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Synonym: Oxiphencycliminum; Manir; Antulcus; Caridan; Naridan; Zamanil; Oxifencicliminum; Oxyphencycliminum; Oxyphencycliminum [INN-Latin]; Daricol; Daricon
IUPAC/Chemical Name: (1-methyl-5,6-dihydro-4H-pyrimidin-2-yl)methyl 2-cyclohexyl-2-hydroxy-2-phenylacetate
InChi Key: DUDKAZCAISNGQN-UHFFFAOYSA-N
InChi Code: InChI=1S/C20H28N2O3/c1-22-14-8-13-21-18(22)15-25-19(23)20(24,16-9-4-2-5-10-16)17-11-6-3-7-12-17/h2,4-5,9-10,17,24H,3,6-8,11-15H2,1H3
SMILES Code: CN1CCCN=C1COC(=O)C(C2CCCCC2)(C3=CC=CC=C3)O
Appearance: Solid powder
Purity: >98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO, not in water
Shelf Life: >2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code: 2934.99.9001
The following data is based on the product molecular weight 344.46 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
|Concentration / Solvent Volume / Mass||1 mg||5 mg||10 mg|
|1 mM||1.15 mL||5.76 mL||11.51 mL|
|5 mM||0.23 mL||1.15 mL||2.3 mL|
|10 mM||0.12 mL||0.58 mL||1.15 mL|
|50 mM||0.02 mL||0.12 mL||0.23 mL|
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