Amidantel free base

    WARNING: This product is for research use only, not for human or veterinary use.

MedKoo CAT#: 524226

CAS#: 49745-00-8 (free base)

Description: Amidantel free base is a new aminophenylamidine with an interesting anthelminthic spectrum. In rodents the compound is active against nematodes, filariae and cestodes. Of special interest is the high efficacy in dogs against hookworms and large roundworms. Amidantel was well tolerated by all animals tested and did not show teratogenic effects.

Chemical Structure

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Amidantel free base
CAS# 49745-00-8 (free base)
Instruction

Theoretical Analysis

MedKoo Cat#: 524226
Name: Amidantel free base
CAS#: 49745-00-8 (free base)
Chemical Formula: C13H19N3O2
Exact Mass: 249.15
Molecular Weight: 249.310
Elemental Analysis: C, 62.63; H, 7.68; N, 16.85; O, 12.84

Price and Availability

This product is not in stock, which may be available by custom synthesis. For cost-effective reason, minimum order is 1g (price is usually high, lead time is 2~3 months, depending on the technical challenge). Quote less than 1g will not be provided. To request quote, please email to sales @medkoo.com or click below button.
Note: Price will be listed if it is available in the future.

Request quote for custom synthesis

Related CAS #: 49745-00-8 (free base)   69884-15-7 (HCl)    

Synonym: Amidantel; Amidantel free base; BAY d 8815; BAY d-8815; BAY d8815; BAYd 8815; BAYd-8815; BAYd8815;

IUPAC/Chemical Name: 4'-((1-(Dimethylamino)ethylidene)amino)-2-methoxyacetanilide

InChi Key: MKFMTNNOZQXQBP-GXDHUFHOSA-N

InChi Code: InChI=1S/C13H19N3O2/c1-10(16(2)3)14-11-5-7-12(8-6-11)15-13(17)9-18-4/h5-8H,9H2,1-4H3,(H,15,17)/b14-10+

SMILES Code: O=C(NC1=CC=C(/N=C(N(C)C)\C)C=C1)COC

Appearance: Solid powder

Purity: >98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility: Soluble in DMSO, not in water

Shelf Life: >2 years if stored properly

Drug Formulation: This drug may be formulated in DMSO

Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code: 2934.99.9001

More Info: Related: 49745-00-8(Amidantel) 69884-15-7 (Amidantel hydrochloride).

Biological target:
In vitro activity:
In vivo activity:

Preparing Stock Solutions

The following data is based on the product molecular weight 249.31 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
Formulation protocol:
In vitro protocol:
In vivo protocol:

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