BIA10-2474
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    WARNING: This product is for research use only, not for human or veterinary use.

MedKoo CAT#: 522618

CAS#: 1233855-46-3

Description: BIA10-2474 is a long-acting reversible inhibitor of fatty acid amide hydrolase (FAAH) that increases levels of the neurotransmitter anandamide in the central nervous system and in peripheral tissues (that is, the rest of the body other than the brain and spinal cord). BIA 10-2474 interacts with the human endocannabinoid system. BIA 10-2474 was in development for the treatment of a range of different medical conditions from anxiety to Parkinson's disease, also for the treatment of chronic pain of multiple sclerosis, cancer, hypertension or the treatment of obesity. A clinical trial with this drug was underway in Rennes, France, in which severe adverse events occurred in January 2016 affecting 5 patients, including leading to the death of one.


Price and Availability

Size
Price

25mg
USD 250
200mg
USD 1250
2g
USD 5450
Size
Price

50mg
USD 450
500mg
USD 1950
5g
USD 8450
Size
Price

100mg
USD 750
1g
USD 3250

BIA 10-2474, purity > 98%, is in stock. Current shipping out time is about 2 weeks after order is received. CoA, QC data and MSDS documents are available in one week after order is received.


Chemical Structure

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Theoretical Analysis

MedKoo Cat#: 522618
Name: BIA10-2474
CAS#: 1233855-46-3
Chemical Formula: C16H20N4O2
Exact Mass: 300.1586
Molecular Weight: 300.362
Elemental Analysis: C, 63.98; H, 6.71; N, 18.65; O, 10.65


Synonym: BIA 10-2474; BIA-10-2474; BIA10-2474.

IUPAC/Chemical Name: 3-(1-(cyclohexyl(methyl)carbamoyl)-1H-imidazol-4-yl)pyridine 1-oxide

InChi Key: DOWVMJFBDGWVML-UHFFFAOYSA-N

InChi Code: InChI=1S/C16H20N4O2/c1-18(14-7-3-2-4-8-14)16(21)19-11-15(17-12-19)13-6-5-9-20(22)10-13/h5-6,9-12,14H,2-4,7-8H2,1H3

SMILES Code: O=C(N1C=C(C2=C[N+]([O-])=CC=C2)N=C1)N(C3CCCCC3)C


Technical Data

Appearance:
Solid powder

Purity:
>98% (or refer to the Certificate of Analysis)

Shipping Condition:
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition:
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility:
Soluble in DMSO, not in water

Shelf Life:
>2 years if stored properly

Drug Formulation:
This drug may be formulated in DMSO

Stock Solution Storage:
0 - 4 C for short term (days to weeks), or -20 C for long term (months).

Harmonized System Code:
293490