WARNING: This product is for research use only, not for human or veterinary use.
MedKoo CAT#: 317504
CAS#: 58-25-3
Description: Chlordiazepoxide is a sedative/hypnotic drug and benzodiazepine. Chlordiazepoxide was the first benzodiazepine to be synthesized and the discovery of chlordiazepoxide was by pure chance. Chlordiazepoxide and other benzodiazepines were initially accepted with widespread public approval but were followed with widespread public disapproval and recommendations for more restrictive medical guidelines for its use. Chlordiazepoxide has a medium to long half-life but its active metabolite has a very long half-life. The drug has amnestic, anticonvulsant, anxiolytic, hypnotic and skeletal muscle relaxant properties. Chlordiazepoxide is discontinued.
MedKoo Cat#: 317504
Name: Chlordiazepoxide
CAS#: 58-25-3
Chemical Formula: C11H12Cl2N2O5
Exact Mass:
Molecular Weight: 323.13
Elemental Analysis: C, 40.89; H, 3.74; Cl, 21.94; N, 8.67; O, 24.76
This product is not in stock, which may be available by custom synthesis.
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Synonym: Chlordiazepoxide; Chlornitromycin; NSC 3069; Chloromycetin; Levomycetin; Chlorocid; Globenicol; Kloramfenikol; Levomycetin; Ophthochlor; Syntomycin;
IUPAC/Chemical Name: 2,2-dichloro-N-[(1R,2R)-1,3-dihydroxy-1-(4-nitrophenyl)propan-2-yl]acetamide
InChi Key: WIIZWVCIJKGZOK-UHFFFAOYSA-N
InChi Code: InChI=1S/C11H12Cl2N2O5/c12-10(13)11(18)14-8(5-16)9(17)6-1-3-7(4-2-6)15(19)20/h1-4,8-10,16-17H,5H2,(H,14,18)
SMILES Code: C1=CC(=CC=C1C(C(CO)NC(=O)C(Cl)Cl)O)[N+](=O)[O-]
Appearance: Solid powder
Purity: >98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO, not in water
Shelf Life: >2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code: 2934.99.9001
The following data is based on the product molecular weight 323.13 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
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