Biperiden Hydrochloride
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MedKoo CAT#: 317328

CAS#: 1235-82-1 (HCl)

Description: Biperiden hydrochloride is a muscarinic antagonist that has effects in both the central and peripheral nervous systems. Biperiden Hydrochloride has been used in the treatment of arteriosclerotic, idiopathic, and postencephalitic parkinsonism. It has also been used to alleviate extrapyramidal symptoms induced by phenothiazine derivatives and reserpine.


Chemical Structure

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Biperiden Hydrochloride
CAS# 1235-82-1 (HCl)

Theoretical Analysis

MedKoo Cat#: 317328
Name: Biperiden Hydrochloride
CAS#: 1235-82-1 (HCl)
Chemical Formula: C21H30ClNO
Exact Mass:
Molecular Weight: 347.92
Elemental Analysis: C, 72.49; H, 8.69; Cl, 10.19; N, 4.03; O, 4.60

Price and Availability

Size Price Availability Quantity
50.0mg USD 350.0 2 Weeks
100.0mg USD 550.0 2 Weeks
200.0mg USD 950.0 2 Weeks
500.0mg USD 1950.0 2 Weeks
1.0g USD 2950.0 2 Weeks
2.0g USD 5250.0 2 Weeks
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Related CAS #: 1235-82-1 (HCl)   514-65-8 (free base).  

Synonym: Akineton; Akinophyl; Akineton hydrochloride; Biperiden; Biperiden Hydrochloride; Biperiden.

IUPAC/Chemical Name: 1-(5-Bicyclo[2.2.1]hept-2-enyl)-1-phenyl-3-(1-piperidinyl)propan-1-ol hydrochloride

InChi Key: RDNLAULGBSQZMP-UHFFFAOYSA-N

InChi Code: InChI=1S/C21H29NO.ClH/c23-21(19-7-3-1-4-8-19,11-14-22-12-5-2-6-13-22)20-16-17-9-10-18(20)15-17;/h1,3-4,7-10,17-18,20,23H,2,5-6,11-16H2;1H

SMILES Code: C1CCN(CC1)CCC(C2CC3CC2C=C3)(C4=CC=CC=C4)O.Cl

Appearance: White to off-white solid powder.

Purity: >98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility: Soluble in DMSO, not in water

Shelf Life: >2 years if stored properly

Drug Formulation: This drug may be formulated in DMSO

Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code: 2934.99.9001

Preparing Stock Solutions

The following data is based on the product molecular weight 347.92 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL

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