Bepridil HCl
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MedKoo CAT#: 317318

CAS#: 68099-86-5 (HCl)

Description: Bepridil Hydrochloride is the hydrochloride salt form of bepridil, a calcium antagonist and class IV anti-arrhythmic agent. Bepridil hydrochloride blocks calcium entry through membranous calcium channels of coronary and peripheral vascular smooth muscle, thereby dilating coronary arteries and peripheral arterioles. This drug is used to treat chronic stable and variant angina pectoris. Bepridil hydrochloride has antihypertensive and selective anti-arrhythmia activities and acts as a calmodulin antagonist.


Chemical Structure

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Bepridil HCl
CAS# 68099-86-5 (HCl)

Theoretical Analysis

MedKoo Cat#: 317318
Name: Bepridil HCl
CAS#: 68099-86-5 (HCl)
Chemical Formula: C24H33ClN2O
Exact Mass:
Molecular Weight: 400.991
Elemental Analysis: C, 71.89; H, 8.30; Cl, 8.84; N, 6.99; O, 3.99

Price and Availability

Size Price Availability Quantity
200.0mg USD 350.0 2 weeks
500.0mg USD 750.0 2 weeks
1.0g USD 1250.0 2 weeks
2.0g USD 2150.0 2 weeks
5.0g USD 4750.0 2 weeks
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Related CAS #: 64706-54-3 (free base)   68099-86-5 (HCl)   74764-40-2 (HCl hydrate)   99239-96-0 (S-isomer HCl)   110143-75-4 (S-isomer)   110143-74-3 (R-isomer)    

Synonym: CERM 1978; CERM-1978; CERM1978; Angopril, Bepadin, Bepridil HCl, Bepridil hydrochloride;

IUPAC/Chemical Name: 1-Pyrrolideneethanamine, beta-((2-methylpropoxy)methyl)-N-phenyl-N-(phenylmethyl)-, hydrochloride

InChi Key: IHYCZMGXKHVACP-UHFFFAOYSA-N

InChi Code: InChI=1S/C24H32N2O.ClH/c1-20(2)18-27-19-22(24-14-9-15-25-24)17-26(23-12-7-4-8-13-23)16-21-10-5-3-6-11-21;/h3-8,10-13,20,22H,9,14-19H2,1-2H3;1H

SMILES Code: CC(C)COCC(C1=NCCC1)CN(C2=CC=CC=C2)CC3=CC=CC=C3.[H]Cl

Appearance: Solid powder

Purity: >98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility: Soluble in DMSO, not in water

Shelf Life: >2 years if stored properly

Drug Formulation: This drug may be formulated in DMSO

Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code: 2934.99.9001

Preparing Stock Solutions

The following data is based on the product molecular weight 400.991 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL

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