WARNING: This product is for research use only, not for human or veterinary use.
MedKoo CAT#: 317353
CAS#: 980-71-2 (maleate)
Description: Brompheniramine, commonly marketed as its salt brompheniramine maleate, is an antihistamine drug of the propylamine (alkylamine) class. It is readily available over the counter and is indicated for the treatment of the symptoms of the common cold and allergic rhinitis, such as runny nose, itchy eyes, watery eyes, and sneezing. It is a first-generation antihistamine. Brompheniramine works by acting as an antagonist of histamine H1 receptors. It also functions as a moderately effective anticholinergic agent, and is likely an antimuscarinic agent similar to other common antihistamines such as diphenhydramine.
MedKoo Cat#: 317353
Name: Brompheniramine maleate
CAS#: 980-71-2 (maleate)
Chemical Formula: C20H23BrN2O4
Exact Mass: 318.07316
Molecular Weight: 435.318
Elemental Analysis: C, 55.18; H, 5.33; Br, 18.36; N, 6.44; O, 14.70
Brompheniramine maleate, purity > 98%, is in stock. Current shipping out time is about 2 weeks after order is received. CoA, QC data and MSDS documents are available in one week after order is received.
Related CAS #: 980-71-2 (maleate) 86-22-6 (free base).
Synonym: Brompheniramine, Bromfed, Dimetapp, Bromfenex, Dimetane, BPN, Lodrane
IUPAC/Chemical Name: 3-(4-bromophenyl)-N,N-dimethyl-3-pyridin-2-ylpropan-1-amine maleate
InChi Key: SRGKFVAASLQVBO-BTJKTKAUSA-N
InChi Code: InChI=1S/C16H19BrN2.C4H4O4/c1-19(2)12-10-15(16-5-3-4-11-18-16)13-6-8-14(17)9-7-13;5-3(6)1-2-4(7)8/h3-9,11,15H,10,12H2,1-2H3;1-2H,(H,5,6)(H,7,8)/b;2-1-
SMILES Code: CN(C)CCC(C1=CC=C(Br)C=C1)C2=NC=CC=C2.O=C(O)/C=C\C(O)=O
The following data is based on the product molecular weight 435.318 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
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antihistamines in inhibition of oxidative burst of professional phagocytes. Gen
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2: Liu YP, Huang TS, Tung CS, Lin CC. Effects of atomoxetine on attention and
impulsivity in the five-choice serial reaction time task in rats with lesions of
dorsal noradrenergic ascending bundle. Prog Neuropsychopharmacol Biol Psychiatry.
2015 Jan 2;56:81-90. doi: 10.1016/j.pnpbp.2014.08.007. Epub 2014 Aug 21. PubMed
PMID: 25151304.