WARNING: This product is for research use only, not for human or veterinary use.
MedKoo CAT#: 317156
CAS#: 2751-68-0
Description: Acetophenazine is discontinued (DEA controlled substance). It is an antipsychotic drug used in the treatment of psychosis. It is also used to treat hallucinations or delusions. It primarily targets the dopamine D2 receptor.
MedKoo Cat#: 317156
Name: Acetophenazine
CAS#: 2751-68-0
Chemical Formula: C23H29N3O2S
Exact Mass: 411.19805
Molecular Weight: 411.56
Elemental Analysis: C, 67.12; H, 7.10; N, 10.21; O, 7.77; S, 7.79
This product is not in stock, which may be available by custom synthesis.
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Synonym: Tindal; Acephenazinum; Acetophenazine.
IUPAC/Chemical Name: 1-[10-[3-[4-(2-hydroxyethyl)piperazin-1-yl]propyl]phenothiazin-2-yl]ethanone
InChi Key: WNTYBHLDCKXEOT-UHFFFAOYSA-N
InChi Code: InChI=1S/C23H29N3O2S/c1-18(28)19-7-8-23-21(17-19)26(20-5-2-3-6-22(20)29-23)10-4-9-24-11-13-25(14-12-24)15-16-27/h2-3,5-8,17,27H,4,9-16H2,1H3
SMILES Code: CC(C(C=C1N2CCCN3CCN(CCO)CC3)=CC=C1SC4=C2C=CC=C4)=O
Appearance: Solid powder
Purity: >98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO, not in water
Shelf Life: >2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code: 2934.99.9001
The following data is based on the product molecular weight 411.56 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
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