WARNING: This product is for research use only, not for human or veterinary use.
MedKoo CAT#: 466175
CAS#: unknown
Description: PSB-16282 is a novel Potent Agonist of the Orphan G Protein-Coupled Receptor GPR17 (EC50 12 nM).
MedKoo Cat#: 466175
Name: PSB-16282
CAS#: unknown
Chemical Formula: C19H24FNO5
Exact Mass: 365.1639
Molecular Weight: 365.4014
Elemental Analysis: C, 62.45; H, 6.62; F, 5.20; N, 3.83; O, 21.89
This product is not in stock, which may be available by custom synthesis.
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Synonym: PSB-16282; PSB16282; PSB 16282; PSB1; PSB 1; PSB-1;
IUPAC/Chemical Name: 3-(2-carboxyethyl)-4-fluoro-6-((5-methylhexyl)oxy)-1H-indole-2-carboxylic acid
InChi Key: LOUBKDFSJXMELF-UHFFFAOYSA-N
InChi Code: InChI=1S/C19H24FNO5/c1-11(2)5-3-4-8-26-12-9-14(20)17-13(6-7-16(22)23)18(19(24)25)21-15(17)10-12/h9-11,21H,3-8H2,1-2H3,(H,22,23)(H,24,25)
SMILES Code: O=C(C(N1)=C(CCC(O)=O)C2=C1C=C(OCCCCC(C)C)C=C2F)O
Appearance: Solid powder
Purity: >98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: To be determined
Shelf Life: >2 years if stored properly
Drug Formulation: To be determined
Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code: 2934.99.9001
The following data is based on the product molecular weight 365.4014 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
1: Braune M, Scherf N, Heine C, Sygnecka K, Pillaiyar T, Parravicini C, Heimrich B, Abbracchio MP, Müller CE, Franke H. Involvement of GPR17 in Neuronal Fibre Outgrowth. Int J Mol Sci. 2021 Oct 28;22(21):11683. doi: 10.3390/ijms222111683. PMID: 34769111; PMCID: PMC8584086.
