PFK-015
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    WARNING: This product is for research use only, not for human or veterinary use.

MedKoo CAT#: 406616

CAS#: 4382-63-2

Description: PFK-015 is a potent inhibitor of PFKFB3. The preliminary results in a U87GM xenograft model have shown that PFK-015 has comparable activity to Temozolomide. PFK-015 inhibits glucoseuptake by tumors.


Chemical Structure

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PFK-015
CAS# 4382-63-2

Theoretical Analysis

MedKoo Cat#: 406616
Name: PFK-015
CAS#: 4382-63-2
Chemical Formula: C17H12N2O
Exact Mass: 260.09496
Molecular Weight: 260.29
Elemental Analysis: C, 78.44; H, 4.65; N, 10.76; O, 6.15

Price and Availability

Size Price Availability Quantity
100.0mg USD 650.0 2 Weeks
200.0mg USD 950.0 2 Weeks
500.0mg USD 1650.0 2 Weeks
1.0g USD 2650.0 2 Weeks
2.0g USD 4650.0 2 Weeks
5.0g USD 7450.0 2 Weeks
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Synonym: PFK015; PFK 015; PFK015.

IUPAC/Chemical Name: (E)-3-(pyridin-3-yl)-1-(quinolin-3-yl)prop-2-en-1-one

InChi Key: LFVHDRPWNYRNLS-BQYQJAHWSA-N

InChi Code: InChI=1S/C17H12N2O/c20-17(8-7-13-4-3-9-18-11-13)15-10-14-5-1-2-6-16(14)19-12-15/h1-12H/b8-7+

SMILES Code: O=C(C1=CC2=CC=CC=C2N=C1)/C=C/C3=CC=CN=C3

Appearance: Solid powder

Purity: >98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility: Soluble in DMSO, not in water

Shelf Life: >2 years if stored properly

Drug Formulation: This drug may be formulated in DMSO

Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code: 2934.99.9001

Preparing Stock Solutions

The following data is based on the product molecular weight 260.29 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL

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PFK-015

100.0mg / USD 650.0


Additional Information