WARNING: This product is for research use only, not for human or veterinary use.
MedKoo CAT#: 576899
CAS#: 134208-17-6
Description: Mazapertine is an antipsychotic agent.
MedKoo Cat#: 576899
Name: Mazapertine
CAS#: 134208-17-6
Chemical Formula: C26H35N3O2
Exact Mass: 421.2729
Molecular Weight: 421.58
Elemental Analysis: C, 74.07; H, 8.37; N, 9.97; O, 7.59
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Synonym: Mazapertine
IUPAC/Chemical Name: (3-((4-(2-isopropoxyphenyl)piperazin-1-yl)methyl)phenyl)(piperidin-1-yl)methanone
InChi Key: ZKZFPRUSWCYSGT-UHFFFAOYSA-N
InChi Code: InChI=1S/C26H35N3O2/c1-21(2)31-25-12-5-4-11-24(25)28-17-15-27(16-18-28)20-22-9-8-10-23(19-22)26(30)29-13-6-3-7-14-29/h4-5,8-12,19,21H,3,6-7,13-18,20H2,1-2H3
SMILES Code: CC(C)Oc1ccccc1N2CCN(Cc3cccc(c3)C(=O)N4CCCCC4)CC2
Appearance: Solid powder
Purity: >98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: To be determined
Shelf Life: >2 years if stored properly
Drug Formulation: To be determined
Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code: 2934.99.9001
The following data is based on the product molecular weight 421.58 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
1. Caldwell GW, Wu WN, McKown LA, Diane Gauthier A, Masucci JA, Jones WJ, Leo GC, Reitz AB. Distribution and metabolism of the antipsychotic agent mazapertine succinate in rats. J Pharm Biomed Anal. 2006 May 3;41(2):500-9. doi: 10.1016/j.jpba.2005.10.052. Epub 2005 Dec 28. PMID: 16386397.
