WARNING: This product is for research use only, not for human or veterinary use.
MedKoo CAT#: 559316
Description: MA-Mlvp is a fluorescent vasopressin analog which are well-suited to the study of renal vasopressin receptors. MA-MLVP at a concentration of 10^(-6) M increased adenylate cyclase activity in canine renal plasma membranes 2.9 times that of basal activity. A maximally active concentration of AVP (1 microM) increased adenylate cyclase activity in canine renal plasma membranes to a value 2.7 times that of basal activity. MA-MLVP at a concentration of 10^(-6) M increased the cAMP content of porcine kidney cells from a basal level of 43 to 160 pmol/mg of cell protein.
MedKoo Cat#: 559316
Chemical Formula: C54H71N13O13S2
Exact Mass: 1173.4736
Molecular Weight: 1174.36
Elemental Analysis: C, 55.23; H, 6.09; N, 15.51; O, 17.71; S, 5.46
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Synonym: Vasopressin; MA-Mlvp; MA Mlvp; MAMlvp
IUPAC/Chemical Name: Vasopressin, 1-(3-mercaptopropanoic acid)-8-(N6-(2-(methylamino)benzoyl)-L-lysine)-
InChi Key: UHHGQCRVKWSIPI-UHFFFAOYSA-N
InChi Code: InChI=1S/C54H71N13O13S2/c1-58-35-13-6-5-12-34(35)47(73)59-23-8-7-14-36(48(74)60-29-45(57)71)63-53(79)42-15-9-24-67(42)54(80)41-30-82-81-25-22-46(72)61-38(27-32-16-18-33(68)19-17-32)50(76)64-39(26-31-10-3-2-4-11-31)51(77)62-37(20-21-43(55)69)49(75)65-40(28-44(56)70)52(78)66-41/h2-6,10-13,16-19,36-42,58,68H,7-9,14-15,20-30H2,1H3,(H2,55,69)(H2,56,70)(H2,57,71)(H,59,73)(H,60,74)(H,61,72)(H,62,77)(H,63,79)(H,64,76)(H,65,75)(H,66,78)
SMILES Code: CNc1ccccc1C(=O)NCCCCC(NC(=O)C2CCCN2C(=O)C3CSSCCC(=O)NC(Cc4ccc(O)cc4)C(=O)NC(Cc5ccccc5)C(=O)NC(CCC(=O)N)C(=O)NC(CC(=O)N)C(=O)N3)C(=O)NCC(=O)N
Appearance: Solid powder
Purity: >98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: To be determined
Shelf Life: >2 years if stored properly
Drug Formulation: To be determined
Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code: 2934.99.9001
The following data is based on the product molecular weight 1174.36 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
|Concentration / Solvent Volume / Mass||1 mg||5 mg||10 mg|
|1 mM||1.15 mL||5.76 mL||11.51 mL|
|5 mM||0.23 mL||1.15 mL||2.3 mL|
|10 mM||0.12 mL||0.58 mL||1.15 mL|
|50 mM||0.02 mL||0.12 mL||0.23 mL|
Lutz WH, Londowski JM, Kumar R. The synthesis and biological activity of four novel fluorescent vasopressin analogs. J Biol Chem. 1990 Mar 15;265(8):4657-63. PMID: 2155234.