WARNING: This product is for research use only, not for human or veterinary use.
MedKoo CAT#: 533068
Description: PA-082 is a Novel partial agonist of peroxisome proliferator-activated receptor-γ (PPARγ), recruiting PPARγ-coactivator-1α, preventing triglyceride accumulation, and potentiating insulin signaling in vitro.
MedKoo Cat#: 533068
Chemical Formula: C33H38N2O5
Exact Mass: 542.2781
Molecular Weight: 542.676
Elemental Analysis: C, 73.04; H, 7.06; N, 5.16; O, 14.74
This product is not in stock, which may be available by custom synthesis.
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Synonym: PA-082; PA 082; PA082
IUPAC/Chemical Name: 1-(3,4-Dimethoxy-benzyl)-6,7-dimethoxy-4-[4-(2-methoxy-phenyl)-piperidin-1-ylmethyl]-iso-quinoline
InChi Key: DJEGOJNHRNRMHS-UHFFFAOYSA-N
InChi Code: InChI=1S/C33H38N2O5/c1-36-29-9-7-6-8-25(29)23-12-14-35(15-13-23)21-24-20-34-28(16-22-10-11-30(37-2)31(17-22)38-3)27-19-33(40-5)32(39-4)18-26(24)27/h6-11,17-20,23H,12-16,21H2,1-5H3
SMILES Code: COC1=CC=CC=C1C2CCN(CC3=CN=C(CC4=CC=C(OC)C(OC)=C4)C5=C3C=C(OC)C(OC)=C5)CC2
Appearance: Solid powder
Purity: >98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO
Shelf Life: >3 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code: 2934.99.9001
The following data is based on the product molecular weight 542.676 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
|Concentration / Solvent Volume / Mass||1 mg||5 mg||10 mg|
|1 mM||1.15 mL||5.76 mL||11.51 mL|
|5 mM||0.23 mL||1.15 mL||2.3 mL|
|10 mM||0.12 mL||0.58 mL||1.15 mL|
|50 mM||0.02 mL||0.12 mL||0.23 mL|