WARNING: This product is for research use only, not for human or veterinary use.
MedKoo CAT#: 565569
Description: CAND1-Cullin1 destabilizer C60 is a novel destabilizer of cand1-cullin1 interaction, inducing a p53-stress response pathway
MedKoo Cat#: 565569
Name: CAND1-Cullin1 destabilizer C60
Chemical Formula: C27H24ClN3O4
Exact Mass: 489.1455
Molecular Weight: 489.956
Elemental Analysis: C, 66.19; H, 4.94; Cl, 7.24; N, 8.58; O, 13.06
This product is not in stock, which may be available by custom synthesis.
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Synonym: CAND1-Cullin1 destabilizer C60; CAND1 Cullin1 destabilizer C60; CAND1-Cullin1-destabilizer-C60
IUPAC/Chemical Name: Methyl 2-[[6-chloro-1-(4-methoxyphenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indole-2-carbonyl]amino]benzoate
InChi Key: QKKLITDYULGDTP-UHFFFAOYSA-N
InChi Code: InChI=1S/C27H24ClN3O4/c1-34-18-10-7-16(8-11-18)25-24-19(21-15-17(28)9-12-23(21)29-24)13-14-31(25)27(33)30-22-6-4-3-5-20(22)26(32)35-2/h3-12,15,25,29H,13-14H2,1-2H3,(H,30,33)
SMILES Code: O=C(OC)C1=CC=CC=C1NC(N(C2C3=CC=C(OC)C=C3)CCC4=C2NC5=C4C=C(Cl)C=C5)=O
Appearance: Solid powder
Purity: >98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO
Shelf Life: >3 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code: 2934.99.9001
The following data is based on the product molecular weight 489.956 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
|Concentration / Solvent Volume / Mass||1 mg||5 mg||10 mg|
|1 mM||1.15 mL||5.76 mL||11.51 mL|
|5 mM||0.23 mL||1.15 mL||2.3 mL|
|10 mM||0.12 mL||0.58 mL||1.15 mL|
|50 mM||0.02 mL||0.12 mL||0.23 mL|
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