WARNING: This product is for research use only, not for human or veterinary use.
MedKoo CAT#: 461680
Description: SA 2572 is a newly synthesized Ca2+ antagonist having a inhibitory effect on the fast Na+ inward channel.
MedKoo Cat#: 461680
Name: SA 2572
Chemical Formula: C32H41ClN2O6S
Exact Mass: 616.2374
Molecular Weight: 617.19
Elemental Analysis: C, 62.27; H, 6.70; Cl, 5.74; N, 4.54; O, 15.55; S, 5.19
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Synonym: SA 2572; SA-2572; SA2572;
IUPAC/Chemical Name: 1-(2-(5-methoxy-2-(4-(methyl(3,4,5-trimethoxyphenethyl)amino)butoxy)phenyl)benzo[d]thiazol-3(2H)-yl)ethan-1-one hydrochloride
InChi Key: AONMOOKWGFXUKH-UHFFFAOYSA-N
InChi Code: InChI=1S/C32H40N2O6S.ClH/c1-22(35)34-26-11-7-8-12-30(26)41-32(34)25-21-24(36-3)13-14-27(25)40-18-10-9-16-33(2)17-15-23-19-28(37-4)31(39-6)29(20-23)38-5;/h7-8,11-14,19-21,32H,9-10,15-18H2,1-6H3;1H
SMILES Code: COC1=C(OC)C(OC)=CC(CCN(CCCCOC2=CC=C(OC)C=C2C3SC4=CC=CC=C4N3C(C)=O)C)=C1.[H]Cl
Appearance: Solid powder
Purity: >98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO
Shelf Life: >3 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code: 2934.99.03.00
The following data is based on the product molecular weight 617.19 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
|Concentration / Solvent Volume / Mass||1 mg||5 mg||10 mg|
|1 mM||1.15 mL||5.76 mL||11.51 mL|
|5 mM||0.23 mL||1.15 mL||2.3 mL|
|10 mM||0.12 mL||0.58 mL||1.15 mL|
|50 mM||0.02 mL||0.12 mL||0.23 mL|
1: Miyawaki N, Furuta T, Shigei T. Electrophysiologic effects of a novel Ca antagonist, SA2572, in isolated rabbit and guinea pig hearts. J Cardiovasc Pharmacol. 1988 Jul;12(1):65-71. PubMed PMID: 2459537.
2: Fujita M, Ota A, Ito S, Yamamoto K, Kawashima Y, Iso T, Iwao J. Synthesis and calcium antagonistic activity of (+)-(R)- and (-)-(S)-3-acetyl-2-[5-methoxy-2-[4-[N-methyl-N-(3,4,5- trimethoxyphenethyl)amino]butoxy]phenyl]benzothiazoline hydrochloride. Chem Pharm Bull (Tokyo). 1990 Apr;38(4):936-41. PubMed PMID: 2379287.