WARNING: This product is for research use only, not for human or veterinary use.
MedKoo CAT#: 596848
Description: Alprenolol tartrate, (S)- is a 5-HT1A antagonist.
MedKoo Cat#: 596848
Name: Alprenolol tartrate, (S)-
Chemical Formula: C19H29NO8
Molecular Weight: 399.44
Elemental Analysis: C, 57.13; H, 7.32; N, 3.51; O, 32.04
This product is not in stock, which may be available by custom synthesis.
For cost-effective reason, minimum order is 1g (price is usually high, lead time is 2~3 months, depending on the technical challenge).
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Synonym: Alprenolol tartrate, (S)-; (S)-Alprenolol tartrate; l-Alprenolol bitartrate;
IUPAC/Chemical Name: (S)-1-(2-allylphenoxy)-3-(isopropylamino)propan-2-ol (2R)-2,3-dihydroxysuccinate
InChi Key: MADUQKMQKQDWJH-CJDDZGJJSA-N
InChi Code: InChI=1S/C15H23NO2.C4H6O6/c1-4-7-13-8-5-6-9-15(13)18-11-14(17)10-16-12(2)3;5-1(3(7)8)2(6)4(9)10/h4-6,8-9,12,14,16-17H,1,7,10-11H2,2-3H3;1-2,5-6H,(H,7,8)(H,9,10)/t14-;1-,2?/m01/s1
SMILES Code: O[C@H](COC1=CC=CC=C1CC=C)CNC(C)C.O=C(O)[C@H](O)C(O)C(O)=O
Appearance: Solid powder
Purity: >98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO
Shelf Life: >2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code: 2934.99.9001
The following data is based on the product molecular weight 399.44 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
|Concentration / Solvent Volume / Mass||1 mg||5 mg||10 mg|
|1 mM||1.15 mL||5.76 mL||11.51 mL|
|5 mM||0.23 mL||1.15 mL||2.3 mL|
|10 mM||0.12 mL||0.58 mL||1.15 mL|
|50 mM||0.02 mL||0.12 mL||0.23 mL|
1: Tong S, Zheng Y, Yan J, Guan YX, Wu C, Lei W. Preparative enantioseparation of β-blocker drugs by counter-current chromatography using dialkyl L-tartrate as chiral selector based on borate coordination complex. J Chromatogr A. 2012 Nov 9;1263:74-83. doi: 10.1016/j.chroma.2012.09.023. Epub 2012 Sep 12. PubMed PMID: 23021635.
2: Hedeland M, Nygård M, Isaksson R, Pettersson C. Cellulases from the fungi Phanerochaete chrysosporium and Trichoderma reesei as chiral selectors in capillary electrophoresis: applications with displacer plugs and sample preconcentration. Electrophoresis. 2000 May;21(8):1587-96. PubMed PMID: 10832892.
3: Bjorvatn B, Neckelmann D, Ursin R. The 5-HT1A antagonist (-)-alprenolol fails to modify sleep or zimeldine-induced sleep-waking effects in rats. Pharmacol Biochem Behav. 1992 May;42(1):49-56. PubMed PMID: 1388278.
4: Taouis M, Berlan M, Montastruc P, Lafontan M. Characterization of dog fat cell adrenoceptors: variations in alpha-2 and beta adrenergic receptors distribution according to the extent of the fat deposits and the anatomical location. J Pharmacol Exp Ther. 1987 Sep;242(3):1041-9. PubMed PMID: 2821223.