Oxatomide

    WARNING: This product is for research use only, not for human or veterinary use.

MedKoo CAT#: 527461

CAS#: 60607-34-3

Description: Oxatomide is an H1 receptor antagonist, possessing antiserotonergic actions.

Chemical Structure

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Oxatomide
CAS# 60607-34-3
Instruction

Theoretical Analysis

MedKoo Cat#: 527461
Name: Oxatomide
CAS#: 60607-34-3
Chemical Formula: C27H30N4O
Exact Mass: 426.24
Molecular Weight: 426.564
Elemental Analysis: C, 76.03; H, 7.09; N, 13.13; O, 3.75

Price and Availability

This product is not in stock, which may be available by custom synthesis. For cost-effective reason, minimum order is 1g (price is usually high, lead time is 2~3 months, depending on the technical challenge). Quote less than 1g will not be provided. To request quote, please email to sales @medkoo.com or click below button.
Note: Price will be listed if it is available in the future.

Request quote for custom synthesis

Synonym: Oxatomide

IUPAC/Chemical Name: 3-[3-(4-Benzhydrylpiperazin-1-yl)propyl]-1H-benzimidazol-2-one

InChi Key: BAINIUMDFURPJM-UHFFFAOYSA-N

InChi Code: InChI=1S/C27H30N4O/c32-27-28-24-14-7-8-15-25(24)31(27)17-9-16-29-18-20-30(21-19-29)26(22-10-3-1-4-11-22)23-12-5-2-6-13-23/h1-8,10-15,26H,9,16-21H2,(H,28,32)

SMILES Code: O=C1N(CCCN2CCN(C(C3=CC=CC=C3)C4=CC=CC=C4)CC2)C5=CC=CC=C5N1

Appearance: Solid powder

Purity: >98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility: Soluble in DMSO

Shelf Life: >2 years if stored properly

Drug Formulation: This drug may be formulated in DMSO

Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code: 2934.99.9001

More Info:

Biological target:
In vitro activity:
In vivo activity:

Preparing Stock Solutions

The following data is based on the product molecular weight 426.56 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
Formulation protocol:
In vitro protocol:
In vivo protocol:

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13: Buyse GM, Goemans N, Henricson E, Jara A, van den Hauwe M, Leshner R, Florence JM, Mayhew JE, Escolar DM. CINRG pilot trial of oxatomide in steroid-naïve Duchenne muscular dystrophy. Eur J Paediatr Neurol. 2007 Nov;11(6):337-40. Epub 2007 Apr 24. PubMed PMID: 17459739.

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