WARNING: This product is for research use only, not for human or veterinary use.

MedKoo CAT#: 526195

CAS#: 117354-64-0

Description: 2-Hydroxysaclofen is a GABA-B antagonist.

Price and Availability




2-Hydroxysaclofen is not in stock, may be available through custom synthesis. For cost-effective reason, minimum 1 gram order is requested. The product will be characterized by NMR, HPLC and MS analysis. Purity (HPLC) is usually >98%. CoA, QC data, MSDS will be provided when product is successfully made. The estimated lead time is 2-3 months. Please send email to sales@medkoo.com to inquire quote.

Chemical Structure


Theoretical Analysis

MedKoo Cat#: 526195
Name: 2-Hydroxysaclofen
CAS#: 117354-64-0
Chemical Formula: C9H12ClNO4S
Exact Mass: 265.0176
Molecular Weight: 265.708
Elemental Analysis: C, 40.68; H, 4.55; Cl, 13.34; N, 5.27; O, 24.09; S, 12.07

Synonym: 2-Hydroxysaclofen

IUPAC/Chemical Name: 3-Amino-2-(4-chlorophenyl)-2-hydroxypropane-1-sulfonic acid


InChi Code: InChI=1S/C9H12ClNO4S/c10-8-3-1-7(2-4-8)9(12,5-11)6-16(13,14)15/h1-4,12H,5-6,11H2,(H,13,14,15)

SMILES Code: O=S(CC(O)(C1=CC=C(Cl)C=C1)CN)(O)=O

Technical Data

Solid powder

>98% (or refer to the Certificate of Analysis)

Shipping Condition:
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition:
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Soluble in DMSO

Shelf Life:
>2 years if stored properly

Drug Formulation:
This drug may be formulated in DMSO

Stock Solution Storage:
0 - 4 C for short term (days to weeks), or -20 C for long term (months).

Harmonized System Code:


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