NaV1.7 Blocker-801

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MedKoo CAT#: 525621

CAS#: 1235403-75-4

Description: NaV1.7 Blocker-801 is a potent NaV1.7 blocker, being 5-10 fold more potent than NaV 1.2 and NaV 1.6.

Price and Availability

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Pricing updated 2020-08-09. Prices are subject to change without notice.

NaV1.7 Blocker-801 is not in stock, may be available through custom synthesis. For cost-effective reason, minimum 1 gram order is requested. The product will be characterized by NMR, HPLC and MS analysis. Purity (HPLC) is usually >98%. CoA, QC data, MSDS will be provided when product is successfully made. The estimated lead time is 2-3 months. Please send email to to inquire quote.

Chemical Structure


Theoretical Analysis

MedKoo Cat#: 525621
Name: NaV1.7 Blocker-801
CAS#: 1235403-75-4
Chemical Formula: C20H15ClF2N6O3S2
Exact Mass: 524.0304
Molecular Weight: 524.9458
Elemental Analysis: C, 45.76; H, 2.88; Cl, 6.75; F, 7.24; N, 16.01; O, 9.14; S, 12.21

Synonym: NaV1.7 Blocker-801

IUPAC/Chemical Name: 4-[2-(2-Azetidin-3-yl-2H-pyrazol-3-yl)-4-chloro-phenoxy]-2,5-difluoro-N-[1,2,4]thiadiazol-5-yl-benzenesulfonamide


InChi Code: InChI=1S/C20H15ClF2N6O3S2/c21-11-1-2-17(13(5-11)16-3-4-26-29(16)12-8-24-9-12)32-18-6-15(23)19(7-14(18)22)34(30,31)28-20-25-10-27-33-20/h1-7,10,12,24H,8-9H2,(H,25,27,28)


Technical Data

Solid powder

>98% (or refer to the Certificate of Analysis)

Shipping Condition:
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition:
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Soluble in DMSO

Shelf Life:
>2 years if stored properly

Drug Formulation:
This drug may be formulated in DMSO

Stock Solution Storage:
0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code:


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