WARNING: This product is for research use only, not for human or veterinary use.
MedKoo CAT#: 530576
Description: 10074-G5 is a c-Myc/Max interaction inhibitor. 10074-G5, similarly to 10058-F4 (#F3680), specifically inhibits this interaction by binding to c-Myc, thus preventing C-Myc specific DNA binding and target genes regulation.
MedKoo Cat#: 530576
Chemical Formula: C18H14N4O3
Exact Mass: 334.335
Molecular Weight: 334.335
Elemental Analysis: C, 64.67; H, 4.22; N, 16.76; O, 14.36
10074-G5, purity > 98%, is in stock. Current shipping out time is about 2 weeks after order is received. CoA, QC data and MSDS documents are available in one week after order is received.
Synonym: 10074-G5; 10074G5; 10074 G5;
IUPAC/Chemical Name: N-([1,1'-biphenyl]-2-yl)-7-nitrobenzo[c][1,2,5]oxadiazol-4-amine
InChi Key: KMJPYSQOCBYMCF-UHFFFAOYSA-N
InChi Code: InChI=1S/C18H12N4O3/c23-22(24)16-11-10-15(17-18(16)21-25-20-17)19-14-9-5-4-8-13(14)12-6-2-1-3-7-12/h1-11,19H
SMILES Code: O=[N+]([O-])C1=CC=C(C2=NON=C21)NC3=CC=CC=C3C4=CC=CC=C4
|Solvent||Max Conc. mg/mL||Max Conc. mM|
|Soluble in DMSO||100.0|
The following data is based on the product molecular weight 334.335 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
|Concentration / Solvent Volume / Mass||1 mg||5 mg||10 mg|
|1 mM||1.15 mL||5.76 mL||11.51 mL|
|5 mM||0.23 mL||1.15 mL||2.3 mL|
|10 mM||0.12 mL||0.58 mL||1.15 mL|
|50 mM||0.02 mL||0.12 mL||0.23 mL|
The c-Myc oncoprotein and its partner Max are intrinsically disordered (ID) monomers that undergo coupled folding and binding upon heterodimerization.