VU 0361737

    WARNING: This product is for research use only, not for human or veterinary use.

MedKoo CAT#: 531331

CAS#: 1161205-04-4

Description: VU 0361737, also known as ML128, is a selective positive allosteric modulator at mGluR-4 (EC50 values are 240 and 110 nM at human and rat receptors respectively).

Chemical Structure

VU 0361737
CAS# 1161205-04-4

Theoretical Analysis

MedKoo Cat#: 531331
Name: VU 0361737
CAS#: 1161205-04-4
Chemical Formula: C13H11ClN2O2
Exact Mass: 262.0509
Molecular Weight: 262.693
Elemental Analysis: C, 59.44; H, 4.22; Cl, 13.49; N, 10.66; O, 12.18

Price and Availability

Size Price Availability Quantity
100.0mg USD 450.0 2 Weeks
200.0mg USD 650.0 2 Weeks
500.0mg USD 1250.0 2 Weeks
1.0g USD 2150.0 2 Weeks
2.0g USD 3850.0 2 Weeks
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Synonym: VU 0361737, VU-0361737, VU0361737; ML128; ML-128; ML 128;

IUPAC/Chemical Name: N-(4-Chloro-3-methoxyphenyl)-2-pyridinecarboxamide


InChi Code: InChI=1S/C13H11ClN2O2/c1-18-12-8-9(5-6-10(12)14)16-13(17)11-4-2-3-7-15-11/h2-8H,1H3,(H,16,17)


Appearance: White to off-white solid powder

Purity: >98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility: Soluble in DMSO

Shelf Life: >2 years if stored properly

Drug Formulation: This drug may be formulated in DMSO

Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code: 2934.99.9001

Preparing Stock Solutions

The following data is based on the product molecular weight 262.693 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL

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VU 0361737

100.0mg / USD 450.0