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BI-7273
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    WARNING: This product is for research use only, not for human or veterinary use.

MedKoo CAT#: 406830

CAS#: 1883429-21-7

Description: BI-7273 is a potent and selective BRD9 inhibitor. BI-7273 may be useful in further exploring BRD9 bromodomain biology in both in vitro and in vivo settings. Selective inhibitors of bromodomain-containing protein 9 (BRD9) may have therapeutic potential in the treatment of human malignancies and inflammatory diseases.


Price and Availability

Size Price Shipping out time Quantity
100mg USD 1250 2 weeks
200mg USD 1750 2 weeks
500mg USD 2450 2 weeks
1g USD 3050 2 weeks
2g USD 5450 2 weeks
5g USD 9950 2 weeks
Inquire bulk and customized quantity
Pricing updated 2020-10-24. Prices are subject to change without notice.

BI-7273, purity > 98%, is in stock. Current shipping out time is about 2 weeks after order is received. CoA, QC data and MSDS documents are available in one week after order is received. Delivery time: overnight (USA/Canada); 3-5 days (worldwide). Shipping fee: from $30.00 (USA); from $45.00 (Canada); from $70.00 (international).


Chemical Structure

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Theoretical Analysis

MedKoo Cat#: 406830
Name: BI-7273
CAS#: 1883429-21-7
Chemical Formula: C20H23N3O3
Exact Mass: 353.1739
Molecular Weight: 353.422
Elemental Analysis: C, 67.97; H, 6.56; N, 11.89; O, 13.58


Synonym: BI-7273; BI 7273; BI7273.

IUPAC/Chemical Name: 4-(4-((dimethylamino)methyl)-3,5-dimethoxyphenyl)-2-methyl-2,7-naphthyridin-1(2H)-one

InChi Key: RBUYFHLQNPJMQM-UHFFFAOYSA-N

InChi Code: InChI=1S/C20H23N3O3/c1-22(2)11-17-18(25-4)8-13(9-19(17)26-5)16-12-23(3)20(24)15-10-21-7-6-14(15)16/h6-10,12H,11H2,1-5H3

SMILES Code: O=C1N(C)C=C(C2=CC(OC)=C(CN(C)C)C(OC)=C2)C3=CC=NC=C13


Technical Data

Appearance:
Solid powder

Purity:
>98% (or refer to the Certificate of Analysis)

Shipping Condition:
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition:
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility:
Soluble in DMSO

Shelf Life:
>2 years if stored properly

Drug Formulation:
This drug may be formulated in DMSO

Stock Solution Storage:
0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code:
2934.99.9001


References

1: Martin LJ, Koegl M, Bader G, Cockcroft XL, Fedorov O, Fiegen D, Gerstberger T,
Hofmann MH, Hohmann AF, Kessler D, Knapp S, Knesl P, Kornigg S, Müller S, Nar H,
Rogers C, Rumpel K, Schaaf O, Steurer S, Tallant C, Vakoc CR, Zeeb M, Zoephel A,
Pearson M, Boehmelt G, McConnell D. Structure-Based Design of an in Vivo Active
Selective BRD9 Inhibitor. J Med Chem. 2016 May 26;59(10):4462-75. doi:
10.1021/acs.jmedchem.5b01865. Epub 2016 Mar 10. PubMed PMID: 26914985; PubMed
Central PMCID: PMC4885110.