Bay-02752

    WARNING: This product is for research use only, not for human or veterinary use.

MedKoo CAT#: 524378

CAS#: 78991-74-9

Description: Bay-02752 is a hypolipidemic drug. It has been demonstrated in rats to inhibit intestinal cholesterol absorption.


Chemical Structure

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Bay-02752
CAS# 78991-74-9

Theoretical Analysis

MedKoo Cat#: 524378
Name: Bay-02752
CAS#: 78991-74-9
Chemical Formula: C31H44N4O2
Exact Mass: 504.35
Molecular Weight: 504.710
Elemental Analysis: C, 73.77; H, 8.79; N, 11.10; O, 6.34

Price and Availability

This product is not in stock, which may be available by custom synthesis. For cost-effective reason, minimum order is 1g (price is usually high, lead time is 2~3 months, depending on the technical challenge). Quote less than 1g will not be provided. To request quote, please email to sales @medkoo.com or click below button.
Note: Price will be listed if it is available in the future.

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Synonym: Bay-02752; Bay 02752; Bay02752;

IUPAC/Chemical Name: 1H-Indole-1-carboxamide, N,N'-1,11-undecanediylbis(2,3-dihydro-2-methyl-

InChi Key: GOJXYVFOLUSEAA-UHFFFAOYSA-N

InChi Code: InChI=1S/C31H44N4O2/c1-24-22-26-16-10-12-18-28(26)34(24)30(36)32-20-14-8-6-4-3-5-7-9-15-21-33-31(37)35-25(2)23-27-17-11-13-19-29(27)35/h10-13,16-19,24-25H,3-9,14-15,20-23H2,1-2H3,(H,32,36)(H,33,37)

SMILES Code: CC1Cc2ccccc2N1C(=O)NCCCCCCCCCCCNC(=O)N3c4ccccc4CC3C

Appearance: Solid powder

Purity: >98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility: Soluble in DMSO, not in water

Shelf Life: >2 years if stored properly

Drug Formulation: This drug may be formulated in DMSO

Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code: 2934.99.9001

More Info:

Biological target:
In vitro activity:
In vivo activity:

Preparing Stock Solutions

The following data is based on the product molecular weight 504.71 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
Formulation protocol:
In vitro protocol:
In vivo protocol:

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1: Laccabue D, Tortoreto M, Veneroni S, Perego P, Scanziani E, Zucchetti M, Zaffaroni M, D'Incalci M, Bombardelli E, Zunino F, Pratesi G. A novel taxane active against an orthotopically growing human glioma xenograft. Cancer. 2001 Dec 15;92(12):3085-92. PubMed PMID: 11753988.

2: Harnett KM, Walsh CT, Zhang LH. Effects of Bay o 2752, a hypocholesterolemic agent, on intestinal taurocholate absorption and cholesterol esterification. J Pharmacol Exp Ther. 1989 Nov;251(2):502-9. PubMed PMID: 2810110.

3: Kritchevsky D, Klurfeld DM. Influence of N,N'-(1,11-undecandiyl) bis (2,3-dihydro-2-methyl-1H-indole-1-carboxamide) (BAY 02752) on gallstone formation and regression in hamsters. Pharmacol Res Commun. 1987 Oct;19(10):679-84. PubMed PMID: 3441483.