Safotibant

    WARNING: This product is for research use only, not for human or veterinary use.

MedKoo CAT#: 319753

CAS#: 633698-99-4

Description: Safotibant, also known as LF-22-0542, is a bradykinin B1 receptor antagonist which was under development for the topical treatment of diabetic macular oedema.


Price and Availability

Size
Price

1g
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10g
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Size
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2g
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20g
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Size
Price

5g
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Safotibant is not in stock, may be available through custom synthesis. For cost-effective reason, minimum 1 gram order is requested. The product will be characterized by NMR, HPLC and MS analysis. Purity (HPLC) is usually >98%. CoA, QC data, MSDS will be provided when product is successfully made. The estimated lead time is 2-3 months. Please send email to sales@medkoo.com to inquire quote.


Chemical Structure

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Theoretical Analysis

MedKoo Cat#: 319753
Name: Safotibant
CAS#: 633698-99-4
Chemical Formula: C25H34N4O5S
Exact Mass: 502.225
Molecular Weight: 502.63
Elemental Analysis: C, 59.74; H, 6.82; N, 11.15; O, 15.92; S, 6.38


Synonym: LF-22-0542; LF22-0542; LF 22-0542; LF-220542; LF220542; LF 220542; Safotibant.

IUPAC/Chemical Name: N-(4-(4,5-dihydro-1H-imidazol-2-yl)benzyl)-2-(2-((4-methoxy-N,2,6-trimethylphenyl)sulfonamido)ethoxy)-N-methylacetamide

SMILES Code: O=C(N(CC1=CC=C(C2=NCCN2)C=C1)C)COCCN(S(=O)(C3=C(C)C=C(OC)C=C3C)=O)C


Technical Data

Appearance:
Solid powder

Purity:
>98% (or refer to the Certificate of Analysis)

Shipping Condition:
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition:
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility:
Soluble in DMSO, not in water

Shelf Life:
>2 years if stored properly

Drug Formulation:
This drug may be formulated in DMSO

Stock Solution Storage:
0 - 4 C for short term (days to weeks), or -20 C for long term (months).

Harmonized System Code:
293490