OB-2

    WARNING: This product is for research use only, not for human or veterinary use.

MedKoo CAT#: 526108

CAS#: 300689-25-2

Description: OB-2 is a novel inhibitor of stomatin-like protein-3 (STOML3) oligomerization that reversibly reduce the sensitivity of mechanically gated currents in sensory neurons and silence mechanoreceptors in vivo.


Price and Availability

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OB-2 is not in stock, may be available through custom synthesis. For cost-effective reason, minimum 1 gram order is requested. The product will be characterized by NMR, HPLC and MS analysis. Purity (HPLC) is usually >98%. CoA, QC data, MSDS will be provided when product is successfully made. The estimated lead time is 2-3 months. Please send email to sales@medkoo.com to inquire quote.


Chemical Structure

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Theoretical Analysis

MedKoo Cat#: 526108
Name: OB-2
CAS#: 300689-25-2
Chemical Formula: C24H20N6OS
Exact Mass: 440.1419
Molecular Weight: 440.525
Elemental Analysis: C, 65.44; H, 4.58; N, 19.08; O, 3.63; S, 7.28


Synonym: OB-2

IUPAC/Chemical Name: 2-(9-Benzyl-9H-1,3,4,9-tetraaza-fluoren-2-ylsulfanyl)-N-(4-methyl-pyridin-2-yl)-acetamide

InChi Key: XAQKHBSJOQTCAV-UHFFFAOYSA-N

InChi Code: InChI=1S/C24H20N6OS/c1-16-11-12-25-20(13-16)26-21(31)15-32-24-27-23-22(28-29-24)18-9-5-6-10-19(18)30(23)14-17-7-3-2-4-8-17/h2-13H,14-15H2,1H3,(H,25,26,31)

SMILES Code: O=C(NC1=NC=CC(C)=C1)CSC2=NN=C3C(N(CC4=CC=CC=C4)C5=C3C=CC=C5)=N2


Technical Data

Appearance:
Solid powder

Purity:
>98% (or refer to the Certificate of Analysis)

Shipping Condition:
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition:
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility:
Soluble in DMSO

Shelf Life:
>2 years if stored properly

Drug Formulation:
This drug may be formulated in DMSO

Stock Solution Storage:
0 - 4 C for short term (days to weeks), or -20 C for long term (months).

Harmonized System Code:
293490


References

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