MedKoo Biosciences: Products

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Approved anticancer agents	Anticancer agents in trials
Anticaner agents in preclinical trials	Anticancer molecular libraries
Other drug agents	Drug intermediates
Bio-reagents and biochemicals

Browse products by name

2-methoxyestradiol (angiogenesis inhibitor)

4-demethylpenclomedine(DMPEN) (alkylation agent)

4SC-202 (HDAC inhibitor)

4SC-203 (multi-target kinase inhibitor)

4SC-205 (human kinesin spindle protein Eg5 inhibitor)

A-443654 (AKT inhibitor)

A-674563 (AKT inhibitor)

A-769662 (AMPK activator)

Abarelix

ABC294640 (sphingosine kinase-2 inhibitor)

Abexinostat (PCI-24781; CRA-024781) (HDAC inhibitor)

ABI-008 (nab-docetaxel)

ABI-009 (nab-rapamycin)

ABI-101 (nab-17AAG)

Abiraterone (androgen biosynthesis inhibitor)

Abiraterone acetate (androgen biosynthesis inhibitor)

ABR-215050 (Tasquinimod) (angiogenic inhibitor)

ABT-199 (BCL inhibitor)

ABT-263 (Novitoclax) (Bcl-2 Inhibitor)

ABT-348 (receptor tyrosine kinase inhibitor)

ABT-510 (angiogenesis inhibitor)

ABT-518 (MMP inhibitor)

ABT-737 (BCL-2 inhibitor)

ABT-751 (Microtubule Inhibitor)

ABT-767 (PARP inhibitor)

ABT-806 (anti-EGFR monoclonal antibody )

ABT-828 (a biologic compound that blocks angiogenesis of cancer cells)

AC480 (BMS-599626) (HER inhibitor)

Acadesine (AMP-activated protein kinase activator)

ACE-041 (an investigational protein therapeutic that inhibits angiogenesis)

Aclarubicin hydrochloride

Acolbifene (selective estrogen receptor modulator)

ACY-1215 (HDAC6 inhibitor)

Acyline (MER104) (GnRH antagonist)

AD-1001 (immunomodulatory therapy)

Adenine

Aderbasib (INCB007839) (sheddase inhibitor)

ADI-PEG20 (arginine deiminase (ADI) formulated with polyethylene glycol)

ADPM06 (PDT photosensitizer)

ADW742 (NVP-ADW742) (IGF-IR inhibitor)

AE-37 (Vaccine)

AEE788 (EGFR, ErbB2, KDR, and Flt-1 inhibitor)

AEG-40826 (HGS-1029) (IAP Inhibitor)

AEG-41174 ( tyrosine kinase inhibitor)

AEW-541 (NVP-AEW541) (IGF-IR inhibitor)

AEZS-108 (AN-152) (LHRH-receptor specified doxorubicin conjugate)

AEZS-112 (ZEN012) (tubulin inhibitor)

AEZS-130 (EP-1572) (growth hormone agonist)

AF802 (CH5424802) (ALK inhibitor)

Afatinib (BIBW-2992 ) (EGFR inhibitor)

Afimoxifene (selective estrogen receptor modulator)

AFM-13 (a bispecific, tetravalent human antibody for Hodgkin Lymphoma.)

AFP-464 (aryl hydrocarbon receptor agonist)

AFX-2 (North American ginseng extract)

AFX-9901 (anti-angiogenic agent)

AG-013 (Trefoil Factor)

AG-1478 (EGFR inhibitor)

AG-24322 (CDK inhibitor)

AG-490 (EGFR and JAK inhibitor)

Agomelatine

AI-850 (cremaphor-free formulation of paclitaxel)

AKR-501 (thrombopoietin receptor agonist)

Alanosine (antimetabolic agent; adenylosuccinate synthetase inhibitor)

ALB-109564 ( tubulin inhibitor; antimitotic agent)

Alendronate sodium

Alendronate sodium (geranyltranstransferase inhibitor)

Alfacalcidol

Alisertib (MLN-8237) (Aurora A kinase inhibitor)

Alitretinoin

Allopurinol Sodium

Almestrone

Almorexant

ALN-VSP (an RNAi therapeutic for the treatment of liver cancers )

ALT-801 (IL-2 recombinant fusion protein)

Altretamine

Alvespimycin (Hsp90 inhibitor)

Alvocidib (Flavopiridol) (CDK inhibitor)

Ametantrone (DNA intercalator)

AMG-208 (c-Met inhibitor)

AMG-319 (PI3 Kinase inhibitor )

AMG-337 (c-Met inhibitor)

AMG-386 (angiopoietin inhibitor, an anti-angiopoietin peptibody)

AMG-780 (anti-angiopoietin antibody )

AMG-820 (antibody that targets c-fms and decreases tumor TAM function)

AMG-888 (antibody that inhibits HER3 oncogenic signaling)

AMG-900 (inhibitor of Aurora kinases A, B, and C.)

Amifostine

Aminoglutethimide

Aminolevulinic Acid

Amonafide dihydrohloride (topoisomerase II inhibitor)

Amonafide malate (AS-1413) (topoisomerase II inhibitor)

AMP423 (cyanoaziridine-derivative)

Amrubicin

Amrubicin (anthracycline; DNA intercalactor; topoisomerase II inhibitor)

Amsacrine

Amsalog (topoisomerase II inhibitor)

Amsilarotene (TAC-101) (oral synthetic retinoid)

Amuvatinib (MP-470) (Multitargeted receptor tyrosine kinase inhibitor)

AN-207 (LHRH doxorubicin conjugate)

AN-2728 (PDE4 inhibitor)

ANA-773 (TLR7 agonist)

Anamorelin (RC1291) (ghrelin receptor agonist)

Anastrozole

Aneustat (OMN54) (mixture of extracts from three commonly used Chinese medicine components; Ganoderma lucidum, Salvia miltiorrhiza and Scutellaria barbata)

Anidulafungin

Annamycin (DNA intercalactor; topoisomerase II inhibitor)

ANX-510 (thymidylate synthase inhibitor)

ANX-514 (docetaxel new formulation)

ANZ-207 (cancer vaccine)

AP-26113 (dual ALK and EGFR inhibitor)

Apatinib (VEGFR inhibitor)

Apaziquone (bioreductive prodrug, hypoxia toxic agent)

APC-100 (androgen antagonist)

APC-200 (ROS inhibitor)

APC-300 (signal transduction inhibitor)

Apixaban

APO-866 (FK866) (NAMPT inhibitor)

Aprepitant

Apricoxib (COX-2 inhibitor)

AR-12 (OSU-03012) (PDK-1 inhibitor)

AR-42 (HDAC inhibitor)

Armodafinil (CNS stimulantor)

ARN-509 (androgen receptor antagonist)

Aroplatin (DNA crosslinking agent)

ARQ-092 (AKT inhibitor)

ARQ-501 ( R1668, beta-lapachone) (DNA damage checkpoint pathway activator)

ARQ-621 (Eg5 inhibitor)

ARQ-736 (BRAF Inhibitor)

ARQ-761 (beta-lapachone prodrug; DNA damage checkpoint pathway activator)

ARRY-300 (MEK inhibitor)

ARRY-380 (HER2 inhibitor)

ARRY-520 (KSP inhibitor)

ARRY-614 (p38 and Tie2 kinase inhibitor)

Arzoxifene (selective estrogen receptor modulators (SERMs))

AS101 (interleukin-10 inhibitor)

AS-605240 (PI3K Inhibitor)

AS703026 (MSC1936369B) (MEK 1/2 inhibitor)

AS703988 (MSC201510B) (MEK 1/2 inhibitor)

Ascomycin

ASP-3026 (ALK inhibitor)

ASP-9521 (17βHSD5 inhibitor)

AT-101(Gossypol acetic acid) (Bcl-2 inhibitor)

AT-13387 (Hsp90 inhibitor)

AT-406 (IAP inhibitor)

AT-7519 (CDK inhibitor)

AT7867 (AKT inhibitor)

AT-9283 (multiple kinase inhibitor)

Ataluren (PTC124) (CFTR-G542X nonsense allele inhibitor)

Atamestane (aromatase inhibitor)

Atazanavir

Atiprimod (STAT3 inhibitor)

ATN-161 (integrin alpha5beta1 inhibitor)

ATN-224 (SOD1 inhibitor)

Atrasentan (ABT-627) (endothelin A receptor antagonist)

AUY-922 (NVP-AUY922, VER-52296) (Hsp90 inhibitor)

AVL-292 (BTK inhibitor)

AVN-944 (VX-944) (IMPDH inhibitor)

Axitinib (VEGFR inhibitor)

Azacitidine

Azathioprine sodium

AZD1152-HQPA (Aurora B inhibitor)

AZD-1208 (pan-PIM kinase inhibitor)

AZD-1480 (JAK2 inhibitor)

AZD-2014 (mTOR inhibitor）

AZD-2461 (PARP inhibitor)

AZD-3514

AZD-4547 (pan-FGFR inhibitor)

AZD-4769 (EGFR tyrosine kinase inhibitor)

AZD-4877 (KSP inhibitor)

AZD-4992

AZD-5363 (PKB/Akt inhibitor)

AZD-5438 (CDK Inhibitor)

AZD-6126 (tubulin Inhibitor)

AZD-6918

AZD-7451 ( TRK inhibitor)

AZD-7762 (checkpoint kinase inhibitor)

AZD-8055 (mTOR inhibitor)

AZD-8330 (ARRY-704)

AZD-8931 (HER1and HER2 inhibitor)

AZM-475271 (Src tyrosine kinase inhibitor)

Bafetinib (INNO-406) (Bcr/Abl inhibitor)

BAL101553 (microtubulin inhibitor)

BAL27862 (microtubulin inhibitor)

Banoxantrone (hypoxia toxic agent)

Barasertib (AZD-1152) (Aurora B inhibitor)

Bardoxolone methyl (RTA402) (antioxidant inflammation modulator)

Batabulin sodium (tubulin inhibitor)

Batimastat (MMP Inhibitor)

BAY 10-00394 ( (CDK inhibitor)

BAY 79-4620 (Antibody–drug conjugate)

BAY 80-6946 (PI3K inhibitor)

BAY 94-9392 (F18 tumor PET imaging agent)

BBI-608 (Cancer cell stemness inhibitor)

BC-819 (a plasmid comprised of the H19 gene regulatory sequences )

Becatecarin (DNA intercalator)

Beclometasone dipropionate (potent glucocorticoid steroid)

Beclomethasone dipropionate

Belinostat (HDAC inhibitor)

Belotecan (camptothecin derivative; topoisomerase I inhibitor)

Bendamustine HCl

Bendamustine HCl (DNA alkylator)

Benoxaprofen

Beraprost (prostacyclin derivative)

Berubicin (topoisomerase II inhibitor; anthracycline derivative)

Besifloxacin

Betamethasone

Betamethasone dipropionate

Bethanechol Chloride

Betulinic acid ( ALS357) (melanoma-specific cytotoxic agent)

Bevonium methylsulfate (also see CG-201) ( hCG inhibitor)

Bexarotene

BEZ235 ( NVP-BEZ235) (PI3K inhibitor)

Bezielle (BZL-101) (extract of plant Scutellaria barbata; apoptosis inducer)

BGC-945 (ONX-0801) (thymidylate synthase inhibitor)

BGJ-398 (pan FGFR kinase inhibitor)

BGT226 (NPV-BGT226) (PI3K inhibitor)

BHQ-880 (Antibody)

BI-2536 (Polo-like kinase 1 inhibitor)

BI-505 (anti-ICAM-1 monoclonal antibody BI-505 )

BI-811283 (Aurora kinase inhibitor)

BI-831266 (temporally not available)

BI-836825 (temporally not available)

BI-847325 (temporally not available)

BI-853520 (focal adhesion kinase inhibitor)

Biapenem

Bicalutamide

BIIB-015 (DM4-conjugated anti-Cripto monoclonal antibody )

BIIB-021 (CNF2024) (HSP90 inhibitor)

BIIB-022 (a human, nonglycosylated IgG4 monoclonal antibody)

BIIB028 (Hsp90 inhibitor)

BIND-014 (PSMA-targeted docetaxel nanoparticles)

Biricodar

BIW-8962 (anti-ganglioside GM2 monoclonal antibod)

BIX02188 (MEK inhibitor)

BIX-02188 (MEK5 inhibitor)

BIX02189 (MEK inhibitor)

BKM-120 (PI3K inhibitor)

Bleomycin sulfate

Blonanserin

BMN-673 (PARP inhibitor)

BMS-275183 (paciltaxel analogue, tubulin inhibitor)

BMS-536924 (IGF-IR kinase inhibitor)

BMS-641988 (androgen receptor (AR) antagonist)

BMS-690514 (VEGFR inhibitor; HER inhibitor)

BMS-754807 (IGF-1R inhibitor)

BMS-777607 (Met tyrosine kinase inhibitor)

BMS-794833 (Met and VEGFR inhibitor)

BMS-833923 (XL-139)

BMS-863233 (XL-413) (CDC7 kinase inhibitor)

BMS-906024 (NOTCH inhibitor)

BMS-911543 (JAK2 inhibitor)

BMS-936558 (an anti-programmed death-1 (MDX-1106))

BMS-936559 (an anti-programmed death-1)

BNC-105 (Vascular disrupting agent, tubulin polymerization inhibitor)

BNC105P (Vascular disrupting agent, tubulin polymerization inhibitor)

Bortezomib

Bosutinib (Abl and Src inhibitor)

BQS-481

Brivanib (VEGFR2 inhibitor)

Brivanib alaninate (VEGFR2 inhibitor)

Brivudin (RP-101)

Brivudine

Brostallicin

BT-062 (Anti-myeloma monoclonal antibody-DM4 immunoconjugate)

BYL719 (PI3K inhbitor)

C31510 (not available)

Cabazitaxel (XRP6258)

Cabazitaxel (XRP-6258 ) (tubulin inhibitor)

Cabozantinib ( XL-184) (VEGFR2, Met, FLT3, Tie2, Kit and Ret inhibitor)

CAL-101 (PI3K inhibitor)

CALAA-01 (siRNA-based cancer drug)

Calcitriol

Canertinib

Canfosfamide

Capecitabine

Capesaris (GTX-758) (estrogen receptor (ER) alpha agonist)

Carbendazim

Carboplatin

Carboquone

Carboxyamidotriazole orotate (CTO)

Carfilzomib (proteasome inhibitor)

Carmofur

Carmustine

Casopitant mesylate

CB-1400 (Not Available)

CBP-501

CC-1088 (selective cytokine inhibitory drug; phosphodiesterase-4 inhibitor)

CC-115 (DNA-PK/TOR kinase inhibitor)

CC-122 (Pleiotropic Pathway Modulator)

CC-223（mTOR inhibitor）

CC-401

CC-8490

CCT128930 (AKT inhibitor)

CCT-137690 (pan-Aurora kinase inhibitor)

CDB-4124

CDX-011 (antibody-drug conjugate).

CDX-1401 (fusion protein / antibody )

Cediranib (AZD2171) (VEGF inhibitor)

Cefoselis sulfate

Cefsulodine sodium

Celastrol (HSP90 inhibitor)

Celecoxib

Cemadotin

CEP-11981 (VEGFR inhibitor)

CEP-18770 (proteasome inhibitor)

CEP-28122 (Anaplastic Lymphoma Kinase inhibitor)

CEP-7055

CEP-9722 (PARP inhibitor)

Cerovive (NXY-059)

Cevipabulin (antimicrotubule agent)

CF-101

CGC-11047 (PG-11047)

CGS-21680 (adenosine A2A receptor agonist)

CH5132799 (PI3K inhibitor)

CH5424802 (ALK inhibitor)

Chelerythrine chloride

Chidamide (CS055; HBI-8000)

CHIR-265 (also see: RAF-265)

CHIR-99021

Chlorambucil

Chlorin E6

CHR-2845 (HDAC inhibitor)

CHR-3996 (HDAC inhibitor)

Chrysophanic acid (EGFR/mTOR pathway inhibitor)

CHS-828 (NAD inhibitor)

CI-1040 (also see: PD184352)

Cilengitide

Cinacalcet

Cipatinib (oral tyrosine kinase inhibitor)

Cisatracurium besylate

Cisplatin

CJ-15161

CKD-516 (microtubulin inhibitor)

CKI27 (RG7304) (MEK inhibitor)

Cladribine

Clobetasol propionate

Clodronate disodium

Clofarabine

CLR-1404

CLT-008 (human myeloid progenitor cells)

CNDO-101

CNTO-95 (a fully human monoclonal IgG1 antibody)

CO-101 (Gemcitabine elaidate; CP-4126) (antimetabolite agent)

CO-1686 (AVL-301) (EGFR inhibitor)

Cordycepin (also see: OVI-123)

CP-547632 (VEGFR-2 inhibitor)

CP-724714 (HER2 inhibitor)

CPI-613 (metabolic inhibitor)

CPX-1 (formulation of Irinotecan + Floxuridine)

CPX-351 (formulation of cytarabine + daunorubicin)

Crenolanib (CP-868596) (PDGFR inhibitor)

Crizotinib (PF-2341066)

Crizotinib (PF-2341066) (tyrosine kinase inhibitor)

CRLX-101

Crolibulin (EPC2407)

CRS-100 [a live-attenuated strain of Listeria monocytogenes (Lm)]

CRS-207 [a weakened (attenuated) form of Listeria monocytogenes]

CST-101 (the native NK-92 cell-line)

CT-011 (a humanized monoclonal antibody (mAb) that modulates the immune response and inhibits tumor growth and the spread of metastases.)

CUDC-101 (HDAC, EGFR and HER2 inhibitor)

Custiren (TV-1001, OCX-011) [a mixed-backbone antisense oligodeoxynucleotide with chemosensitizing properties.]

CV9103 (mRNA-derived prostate cancer vaccine)

CVT-6883 (A2B adenosine antagonist)

CWP232291 (Wnt signaling inhibitor)

CX-5461 (RNA polymerase I Inhibitor)

CYC-116 (Aurora kinase/VEGFR2 inhibitor)

Cyclophosphamide

Cyproterone acetate

CYT-107 (Interleukin-7)

CYT-387 (JAK inhibitor)

CYT-6091 (a nanotherapeutic manufactured by covalently linking tumor necrosis factor-a (TNF) onto the surface of 30 nm particles of pegylated colloidal gold)

Cytarabine

D-3263

Dabigatran Etexilate

Dabrafenib (GSK-2118436) (B-RAF inhibitor)

Dacarbazine

Dacinostat (NVP-LAQ824)

Dacomitinib (PF-00299804) (EGFR inhibitor)

Dactinomycin

Danoprevir

Danusertib (PHA-739358) (Aurora kinase inhibitor)

Daptomycin

Darinaparsin (ZIO-101)

Darunavir

Dasatinib

Daunorubicin

DCC-2036 (BCR-ABL inhibitor)

Debio-0932 (CUDC-305) (Hsp90 inhibitor)

Dexrazoxane Hydrochloride

Dinaciclib (SCH-727965, PS-095760) (CDK inhibitor)

DJ-927 (Tesetaxel )

DMPEN(4-demethylpenclomedine) (alkylation agent)

Docetaxel

Docosahexaenoic acid

Dofequidar

Doramapimod (p38 MAPK inhibitor)

Dorzolamide hydrochloride

Dovitinib (TKI-258, CHIR258) (fibroblast growth factor receptor 3 (FGFR3) inhibitor)

Doxercalciferol

Doxifluridine

Doxorubicin Hydrochloride

Dromostanolone Propionate

Droxinostat (HDAC inhibitor)

DS-2248

DS-7423 (PI3K/mTOR kinase inhibitor)

Dutasteride

E-3810 (VEGFR/FGFR dual kinase inhibitor)

E6201 ( MEK-1/MEKK-1 inhibitor)

E7016 (PARP inhibitor)

E7050 ( c-Met/VEGFR kinase inhibitor)

E7272 (also see : ONTAK or denileukin diftitox)

E7820 (angiogenesis inhibitor)

EC-20 (tumor imaging agent)

ECC-33 (RG7686) [monoclonal antibody]

Edatrexate

Edotecarin (PHA-782615; J-107088; ED-749) (topoisomerase inhibitor)

Efaproxiral (radiosensitizer)

Eflornithine (CPP-1X)

EGEN-001 [non-viral vector consisting of a plasmid DNA encoding the human gene for interleukin 12 (IL-12)]

EGEN-002 [not available]

Elacridar (P-glycoprotein inhibitor)

Elacytarabine (antimetabolite agent)

Elagolix ( NBI-56418)

Elesclomol (HSP-90 Inhibitor)

Elinafide (DNA intercalator)

Elisidepsin (PM-02734)

Elomotecan (BN-80927) (topoisomerase inhibitor)

Elsamitrucin (DNA intercalator)

Eltrombopag

Eltrombopag (thrombopoietin receptor agonist)

EMD-1204831 (c-MET inhibitor)

EMD-1214063 (c-Met inhibitor)

Eniluracil (dihydropyrimidine dehydrogenase inhibitor)

ENMD-1198 (antimitotic agent)

ENMD-2076 (Aurora kinase inhibitor)

Entecavir

Entinostat (MS-275, SNDX-275) (HDAC inhibitor)

Enzastaurin (LY317615) (protein kinase C beta inhibitor)

EP-100 [an LHRH receptor-targeting ligand conjugated to a novel
membrane-disrupting peptide called CLIP 71.]

Epirubicin hydrochloride

Epofolate (BMS-753493) (folate receptor-targeting antimitotic agent)

Epothilone D ) (tubulin inhibitor)

Eribulin mesylate (E7389)

Eribulin mesylate (E7389) (tubulin inhibitor)

Erismodegib (LDE225, NVP-LDE225) (Smo antagonist)

Erlotinib Hydrochloride

Ertapenem sodium

ES285

Estramustine phosphate sodium

Estriol

Estrone

Etalocib (LY293111) (LTB4 receptor antagonist)

Ethinyl Estradiol

Exatecan (topoisomerase inhibitor)

Exemestane

Exherin

Exisulind

Ezatiostat (glutathione S-transferase P1-1 (GSTP1-1) inhibitor)

EZN-2208 (Pegylated SN-38)

Fenretinide (RAR agonist)

Fludarabine phosphate

Flumethasone

Fluorogestone acetate

Fluorometholone acetate

Fluorouracil

Flutamide

Foretinib (XL880, SK1363089, GSK089, EXEL-2880) (MET/VEGFR2 inhibitor)

Fosaprepitant (antiemetic agent)

Fosbretabulin (combretastatinA-4phosphate, CA4P) (vascular disrupting agent)

Fostamatinib (R788) (Syk kinase inhibitor)

Fotemustine

FT-1050 (Stem Cell Modulator)

Fulvestrant

Galeterone (TOK-001)

Ganciclovir

Ganetespib (STA-9090) (Hsp90 inhibitor)

GANT58 (Hedgehog inhibitor)

GDC-0032 (PI3K inhibitor)

GDC-0068 (AKT inhibitor)

GDC-0152 (IAP inhibitor, Smac mimetic)

GDC-0425 (RG7602) (ChK-1 inhibitor)

GDC-0623 (MEK inhibitor)

GDC-0879 (B-Raf Inhibitor)

GDC-0917 (IAP inhibitor)

GDC-0941 (PI3K inhibitor)

GDC-0973 (XL518) (MEK inhibitor)

GDC-0980 (RG7422) ( PI3 kinase/mTOR inhibitor)

Gefitinib

Gemcitabine Hydrochloride

GENZ-644282

GFB-204 (VEGFR and PDGFR inhibitor)

GGTI-2418 (geranylgeranyltransferase I inhibitor)

GI-4000 (Targeted Molecular Immunogen)

GI-6207 (vaccine)

Gimatecan (topoisomerase inhibtor)

Ginsenoside Rb1

Ginsenosides Ro

Givinostat (ITF2357) (HDAC inhibitor)

GLPG0187 (integrin receptor antagonist)

Glufosfamide

Glutathione

Glyciphosphoramide

Glyfosfin

GO-203-2C (MUC1-targeted peptide)

Golotimod

Goserelin Acetate

Gossypol (Bcl-2 inhibitor)

GPI-15427

GPX100 (anthracycline, DNA intercalator)

GPX150 (anthracycline, DNA intercalator)

Granisetron hydrochloride

GRN-1005 (ANG-1005) (paclitaxel conjugate, microtube inhibitor)

GS-9219

GSK-1059615 (mTOR inhibitor）

GSK-1070916

GSK-1070916A

GSK-1292263 (GPR119 receptor agonist )

GSK-1904529a (IGF-1R Inhibitor)

GSK-2110183 (AKT inhibitor)

GSK-2126458 (PI3K inhibitor, mTOR inhibitor)

GSK-2141795 (Akt inhibitor)

GSK-2256098

GSK-2401502

GSK-2586881 (APN01)

GSK-2636771 (PI3K inhibitor)

GSK-461364 (PLK Inhibitor)

GSK-690693 (pan-Akt kinase inhibitor)

Gusperimus (immunosuppressant agent)

GW788388 (TGF-beta inhibitor)

HA14-1

Halobetasol propionate

HE-3235

Henatinib (multitargeted tyrosine kinase inhibitor)

Heptaplatin

Hesperadin

Hexyl 5-aminolevulinate

Histrelin Acetate

HM30181 (MDR1 inhibitor)

HM781-36B (irreversible pan-HER inhibitor)

HMN-176 (PLK-1 inhibitor)

HMN-214 (PLK-1 inhibitor)

HQK-1004

HSP-990 (HSP inhibitor)

Hycanthone (Topoisomerase inhibitor, DNA intercalator)

Hydroxytyrosol

Hypothemycin

Iboctadekin (immunostimulatory cytokine )

Ibutamoren

Icotinib (EGFR inhibitor)

Imetelstat (GRN-163L)

Imexon (caspase inhibitor)

IMGN-388 (Targeted Antibody Payload, TAP)

IMGN-901 (lorvotuzumab mertansine)

Imidazoacridone

IMO-2055 (EMD1201081)

INC280 (INCB-028060) (c-MET inhibitor, RTK inhibitor)

INCB-24360

Incyclinide

Indibulin (ZIO-301) (tubulin inhibitor)

Indisulam (carbonic anhydrase inhbitor)

Ingenol Mebutate (PEP005)

Iniparib (BSI-201) (PARP inhibitor)

INK-1117 (PI3K inhibitor)

INK-128 (mTOR inhibitor)

INNO-206 (DNA intercalating agent)

INO-1001

Inolitazone (CS-7017, Efatutazone )

INSM-18

Iobenguane

Ioflubenzamide I-131 (MIP-1145)

IPH-2101 (human anti-NK-cell inhibitory receptor mAb)

IPI-145 (INK-1197) (PI3K inhibitor)

IPI-269609 (Hedgehog pathway inhibitor)

IPI-493

IPI-926 (Hedgehog pathway inhibitor)

Irinotecan Hydrochloride

Irofulven

Irosustat (STX64, BN83495)

Isatoribine (toll-like receptor 7 (TLR-7) agonist)

ISF-35 (vaccine)

Iso-Fludelone (microtubulin inhibitor)

Ispinesib

Istradefylline

Ixabepilone

Ixazomib (MLN-9708) (the first oral proteasome inhibitor)

JI-101

JNJ-26481585 (HDAC inhibitor)

JNJ-26483327

JNJ-38877605 (tyrosine kinase inhibitor)

JNS002 (Pegylated liposomal doxorubicin)

JX-594 (thymidine kinase-deleted vaccinia-hGM-CSF)

JX-929 (A highly tumor-selective vaccinia virus )

Kahalalide F

Karenitecin (Cositecan, BNP-1350).

KB-004 (Humaneered™ monoclonal antibody)

Ketamine

KHK-2866 (Anti-HB-EGF Antibody)

KOS-1584 (R1645)

KP372-1 (Akt inhibitor)

KRN5500

KRN7000 (RGI-2001) (immunomodulator)

KRP-203 (Sphingosine-1-phosphate receptor agonist)

KRX-0402

KRX-0601(also see UCN-01)

KU-0063794 (mTOR inhibitor)

KU-55933

KW-2449

KW-2478 (Hsp90 inhibitor)

KX2-391 (rc kinase inhibitor)

Laromustine(VNP40101M)

Larotaxel (XRP9881)

Lasofoxifene

LCL-161

LDK-378 (ALK inhibitor)

LDN-193189

LE-DT (Liposome Encapsulated Docetaxel)

LEE-011

Lemuteporfin (QLT-0074) (PDT photosensitizer)

Lenalidomide

lenvatinib (E7080)

LEP-ETU (liposomal paclitaxel, PNU-93914)

Levamisole Hydrochloride

Levocetirizine

Levoleucovorin Calcium

lexibulin (CYT997) (Vascular disrupting agent)

LGD-4665

LGH447

LGK-974

LGX818 (Raf kinase inhibitor)

Linifanib ( ABT869) (RTK inhibitor)

Linsitnib (OSI-906) (IGF-1R inhibitor)

Lisdexamfetamine dimesylate

Litronesib (aslo see: LY2523355)

Lobaplatin

Lomeguatrib

Lomustine

Lonafarnib (farnesyl transferase inhibitor)

LOR-253 (MTF-1 inhibitor)

LOR-500 (MELK inhibitor)

LP-261

Lucanthone (Topoisomerase inhibitor, DNA intercalator)

Lurtotecan (OSI-221; NX221) (topoisomerase I inhibitor)

LW6 (HIF-1α inhibitor)

LY2090314 (GSK-3 inhibitor)

LY2157299 (TGF-βR inhibitor)

LY2181308 (antisense oligonucleotide)

LY2228820 (p38MAPK inhibitor)

LY2334737 (antimetabolite agent)

LY2584702

LY2603618 (CHK2 inhibitor)

LY2606368

LY2624587 (not available)

LY2780301 (AKT inhibitor)

LY2801653 (c-MET inhibitor)

LY2874455 (FGFR inhibitor)

LY2875358 (anti-c-MET monoclonal antibody)

LY294002 (PI3K inhibitor)

LY2940680

LY3007113 (p38 MAPK inhibitor)

LY475776 (P-glycoprotein inhibitors)

M40403

Marimastat (BB-2516)

Marizomib (NPI-0052) (proteasome inhibitor)

Masitinib (AB1010) (tyrosine kinase inhibitor)

Masoprocol (NDGA) (lipoxygenase inhibitor)

Maytansine (microtubule inhibitor)

MB07133

MDV3100 (selective androgen receptor modulator)

ME-143 (NV-143) (NADH oxidase inhibitor)

ME-344 (mTOR1/2 kinase inhibitor)

Mechlorethamine Gel

Mechlorethamine Hydrochloride

Megestrol Acetate

MEK-162 (ARRY-162) (MEK1/2 inhibitor)

Melphalan Hydrochloride

Meprednisone

Methoxyamine (TRC102) (DNA base excision repair (BER) inhibitor)

Methyl aminolevulinate

Methyl aminolevulinate (PDT photosensitizer)

Methylene Blue

Methylisoindigotin

Methylprednisolone acetate

MG-516 (multi-targeted kinase inhibitor)

MGCD-265 (multitargeted tyrosine kinase inhibitor)

Midostaurin (PKC412)

Mifamurtide

Mifamurtide (L-MTP-PE. MTP-PE) (immunomodulatory agent)

Mifepristone

Milataxel

Milciclib (PHA-848125) (CDK inhibitor and TRKA inhibitor)

Miltefosine

Minoxidil

MINT-1526A (An anti-murine integrin α5β1 antibody)

Mitoxantrone hydrochloride

MK-0429 (ανβ3 Integrin Inhibitor)

MK-0731 (KSP inhibitor)

MK-0752 (notch inhibitor)

MK-1496 (Polo-like kinase 1 inhibitor)

MK-1775 (WEE inhibitor)

MK-2206 (Akt inhibitor)

MK-2461 (Multitargeted Kinase Inhibitor)

MK-4101 (not available)

MK-4827 (PARP inhibitor)

MK-5108 (VX-689)

MK-5172 (protease inhibitor)

MK-8033 (c-MET inhibitor)

MK-8245 (a stearoyl-CoA desaturase (SCD) inhibitor)

MKC-1

MKC1106-PP (immunotherapy)

MKI-833

MLN-2238 (oral proteasome inhibitor, metabolite of MLN9708)

MLN-2480 (Raf kinase inhibitor)

MLN-4924

MLN-8054 (aurora kinase inhibitor)

MM-111 (a bispecific antibody)

MM-151 (EGFR inhibitor)

MM-302 (doxorubicin nanotherapy)

MM-398 (irinotecan nanotherapy)

MN-201

Mocetinostat (MGCD-0103) (HDAC inhibitor)

Mometasone furoate

Motesanib (AMG-706) (tyrosine kinase inhibitor)

Motexafin gadolinium (PDT photosensitizer, radiosensitizer)

Motexafin lutetium (PDT photosensitizer, radiosensitizer)

Moxifloxacin HCl

MP-412 (AV-412) (EGFR/HER2 tyrosine kinase inhibitor)

MPC-2130

MPC-3100 (Hsp90 inhibitor)

MRX-1024

MSX-122

MT-110 (a Bispecific T cell Engager (BiTE)® antibody)

Mubritinib (TAK-165) (EGFR inhibitor)

Muparfostat (PI88, heparin sulfate)

MVA-5T4 (attenuated modified Vaccinia Ankara virus)

Neratinib (HKI272) (HER2 and EGFR inhibitor)

Nilotinib

Nilotinib (Bcr-Abl inhibitor)

Nilutamide

Nimustine

Nintedanib ( BIBF-1120) (VEGFR inhibitor)

Nitroarginine (NG-nitro-L-arginine) (nitric oxide synthase inhibitor)

NK-012 (SN-38-PEG conjugate, camptotecin conjugate)

NKP-1339 (ruthenium-based transferrin targeting agent)

NKP-2235 (gallium-based small molecule)

NKTR-102

NKTR-105

NM-3 (isocoumarin)

NMS-1116354 (CDC7 kinase inhibitor)

NMS-1286937 (PLK1 inhibitor)

Nocodazole

Nolatrexed

Norepinephrine

Noscapine (also see CB-3304)

NOV-002 (chemoprotective agent)

Novitoclax (ABT-263) (Bcl-2 Inhibitor)

NRX-4204

NS-018 (JAK2/Src inhibitor)

NTX-10 (vaccine)

NV-1020 (oncolytic herpes simplex virus type 1)

NV-128 (mTOT inhibitor)

NVP-AEW541 ( AEW541)

NVP-BEP800 (BEP800) (Hsp90 inhibitor)

Obatoclax ( GX15-070) (BCL-2 Inhibitor)

Oblimersen (bcl-2 antisense oligodeoxynucleotide G3139)

OBP-301 (Telomerase-Specific Replication-Competent Adenovirus)

Octreotide

OCV-501

OCX-011 (Custiren, TV-1001) [a mixed-backbone antisense oligodeoxynucleotide with chemosensitizing properties.]

Odanacatib (MK-0822) (protease inhibitor)

ODM-201

Oglufanide

OGX-427 (Hsp27 antisense oligonucleotide )

Olaparib (AZD-2281) (PARP inhibitor)

Oleandrin (PBI-05204)

Omacetaxine mepesuccinate (Homoharringtonine)

Ombrabulin (AVE8062) (tubulin inhibitor)

Omtriptolide

ON-013105

Ondansetron hydrochloride

ONT-093 (OC144-093)

ONX 0805 (SB1578)

ONX-0912 (proteasome inhibitor)

ONX-0914 (immunoproteasome inhibitor)

OPB-31121 (STAT3 inhibitor)

OPB-51602 (STAT3 inhibitor)

Ortataxel

Orteronel (TAK-700) (steroid 17alpha-monooxygenase inhibitor)

OSI-027 (mTOR inhibitor)

OSI-420 (CP-473420) ( EGFR inhibitor )

OSI-7904L(also see: GS7904L, OVI-237 )

OSI-906 (Linsitnib) (IGF-1R inhibitor)

OSI-930

Ostarine (MK-2866, GTX-024)

Oxaliplatin

OXi-4503

Ozarelix (also see: SPI-153)

P2045

P276-00 (DCK inhibitor)

PA799 (PI3K class I inhibitor)

Paclitaxel

Pacritinib (SB1518)

Padeliporfin (WST11, Stakel) (PDT photosensitizer)

Padoporfin (Tookad) (PDT photosensitizer)

Palifosfamide (ZIO-201)

Palomid 529 (PI3K inhibitor; Akt inhibitor; mTOR inhibitor)

Palonosetron hydrochloride

Pamidronate Disodium

Panobinostat (NVP-LBH589; LBH589) (HDAC inhibitor)

Pasireotide (SOM-230) ( somatostatin receptor agonist)

Patupilone (EPO906)

Pazopanib (GW786034) (tyrosine kinase inhibitor )

Pazopanib Hydrochloride (GW786034)

PCI-27483 (factor VIIa inhibitor)

PCI-32765 (BTK inhibitor)

PD-0325901 (MEK inhibitor)

PD-0332991 (CDK Inhibitor)

PD098059 (MEK inhibitor; MAP kinase inhibitor)

PD-153035 (EGFR inhibitor)

Pelitinib (EKB569) (pan-ErbB tyrosine kinase inhibitor)

Pelitrexol (GARFT inhibitor) (glycinamide ribonucleotide formyltransferase)

Peramivir

Perifosine (AKT Inhibitor)

PF-03084014

PF-0337210

PF-03446962 (anti-ALK-1 monoclonal antibody)

PF-03732010 (antibody drug, p-cadherin antagonist)

PF-03758309 (PAK4 inhibitor)

PF-04217903 ( MET tyrosine kinase inhibitor)

PF-04449913

PF-04554878 (FAK inhibitor)

PF-04605412 (anti-A5B1 integrin monoclonal antibody )

PF-04691502 (PI3K/mTOR inhibitor)

PF-0477736

PF-04856884 (CVX-060) [the fusion of two Ang2 sequestering peptides]

PF-0562271 (PF-562271; PF-00562271) (a FAK inhibitor)

PF-3845 (a FAAH Inhibitor)

PHA-665752 (c-MET inhibitor)

Phenoxodiol

Photochlor (PDT photosensitizer)

PHT-427 (Akt inhibitor)

PHY-906

PI-103 (PI3K inhibitor, and mTOR inhibitor)

Picoplatin

Picropodophyllin (AXL1717) (IGF-1 receptor inhibitor)

PIK-75 (PI3K inhibitor)

Pimavanserin

Piroxantrone (topoisomerase II inhibitor)

Pixantrone

PKI-587 (PF-05212384)

Plerixafor

Plevitrexed (BGC-9331)

Plicamycin

Plinabulin (NPI-2358)

Plitidepsin (Aplidine)

PLX-3397 (multitargeted tyrosine kinase inhibitor)

PLX-4720 (B-Raf inhibitor)

PNT-2258 (an oligonucleotide therapeutic encapsulated within a SMARTICLES formulation).

PNU-93914 (liposomal paclitaxel, LEP-ETU)

POL6326 (CXCR4 inhibitor)

Polymyxin B sulphate

Polyphenon E

Pomalidomide

Ponatinib (AP-24534) (tyrosine kinase inhibitor)

Porfimer Sodium

Porfiromycin

PP242 (mTOR inhibitor)

PP-242 (mTOR inhibitor)

PPI-2458

PR-104

Pracinostat (SB939) (HDAC inhibitor)

Pralatrexate

Pralatrexate (dihydrofolate reductase inhibitor)

Prasugrel

Prednimustine

PRI-724 (CBP/beta-catenin antagonist; Wnt signaling pathway inhibitor)

Prinomastat

PRLX-93936

Procarbazine Hydrochloride

PRT-062607

Prucalopride

PRX-302 (protein drug)

PTC-299 (VEGF inhibitor)

Pterostilbene

PTI-188 (a radiolabeled murine anti-melanin antibody)

PU-H71 (Hsp90 inhibitor)

PV-10

PWT33597 (PI3K inhibitor)

PX-12

PX-478 (HIF-1alpha inhibitor)

PX-866 (PI3K inhibitor)

Pyropheophorbide derivatives

Pyroxamide

PZP115891

QBI-139 (protein drug)

Quarfloxin (CX-3543) (G-quadruplex-interactive agent)

Quinacrine (Mepacrine ; CBLC102)

Quinagolide (D2 receptor agonist)

Quinagolide hydrochloride

Quizartinib (AC220) (FLT3 inhibitor)

R1530 (Mitosis-angiogenesis inhibitor)

R306465

R547

R763 (AS703569) (Aurora kinase inhibitor)

Raloxifene

Raltegravir

Raltitrexed

Ramelteon

Ramoplanin

Ranimustine

RC3095

RDEA-436 (MEK inhibitor)

Refametinib (RDEA119; BAY86-9766) (MEK inhibitor)

Regorafenib (BAY 73-4506) (oral multi-kinase inhibitor)

Relacatib

Resiquimod (Toll-like receptor (TLR) agonist)

Resminostat (4SC-201) (HDAC inhibitor)

Resveratrol

Resveratrol(RM1812 , SRT-501)

Retapamulin

Retaspimycin (IPI504) (HSP90 inhibitor)

Retigabine

RG-7167 (MEK inhibitor)

RG-7347 (MNRP1685, R7347, Anti-NRP1)

RG7593 (anti-CD22-MCC-MMAE)

RG7594 (antibody drug)

RG7686 (ECC-33) [monoclonal antibody]

RH1

Ridaforolimus (Deforolimus)

Rigosertib（ON-01910 ) (PLK1 inhibitor)

Rindopepimut (immunotherapy, vaccine)

Riociguat

Rivaroxaban

RM1812 (resveratrol, SRT-501)

RO4929097 (R4733) (gamma-secretase/Notch signalling pathway inhibitor)

RO4987655 (MEK inhibitor)

RO5045337 ( RG7112, R7112) (MDM2 (human homolog of double minutes-2; HDM2) antagonist)

RO5126766 (Raf/MEK dual kinase inhibitor)

RO518426 (V600E BRAF Blocker)

RO5212054 (PLX3603, RG-7256) (BRAF(V600E) kinase inhibitor)

RO5503781 (MDM2 antagonist)

Roflumilast

Rostaporfin (PDT photosensitizer)

RRX-001 (radiosensitizer)

Rubitecan

Rucaparib (PF-01367338, AG-14699) (PARP1 inhibitor)

Rufinamide

Ruxolitinib (INC-424; INCB-18424) (JAK1 inhibitor)

Ruxolitinib (JAK1 inhibitor)

RX-0201 (Akt antisense oligonucleotide)

S31-201

Sabarubicin (DNA intercalator)

Sagopilone (ZK epothilone)

Salirasib

Sapacitabine

SAR103168

SAR256212 (MM-121, human monoclonal antibody)

SAR307746 (REGN901, anti-ANG2 monoclonal antibody)

SAR3419

SAR411298 (FAAH inhibitor. Cancer pain)

Saracatinib (AZD-0530) (Src and Abl inhibitor)

Sardomozide

Sarsasapogenin

Satraplatin

Saxagliptin

SB-1518 (JAK2 inhibitor)

SB202580 (MEK inhibitor; MAP kinase inhibitor)

SB-216763 (glycogen synthase kinase-3 (GSK-3) inhibitor)

SB-431542 (TGF-beta receptor inhibitor, ALK inhibitor)

SB-743921 (KSP inhibitor)

SCH900353

SCH900776 (Chk1 inhibitor)

Seliciclib (CDK inhibitor)

Selumetinib (AZD-6244) (MEK 1/2 inhibitor)

Serdemetan (JNJ-26854165)

SF1126

SGI-110

SGI-1776 (pan-Pim protein kinase inhibitor)

SGN-75 (anti-CD70 monoclonal antibody)

SGX-523 (Met Inhibitor)

SHP-141 (HDAC inhibitor)

Silatecan (AR-67; DB-67) (topoisomerase I inhibitor; camptotecin derivative)

Silibinin ( extract of the milk thistle seeds; mixture of flavonolignans)

Silmitasertib (CX-4945) (CK2 inhibitor)

SJG-136 (BN2629, SG2000) (DNA replication inhibitor)

SL-401 (human IL3 recombinantly conjugated to diphtheria toxin).

SN-2310 (SN-38 conjugate with VE; topoisomerase I inhibitor)

SNS-032 (BMS-387032) (CDK inhibitor)

SNS-314 (Aurora kinase inhibitor)

SNX-2112 (HSP90 inhibitor)

SNX-5422 (PF-4929113)

Soblidotin (tubulin polymerization inhibitor)

Sonoflora 1 ( SF1) (PDT photosensitizer)

Sorafenib

Sotatercept (ACE-011, human fusion protein )

Sotrastaurin (AEB071) (PCK inhibitor)

SPI-1005 (ebselen-containing oral capsule)

SPI-1620

Squalamine

SR13668 (Akt inhibitor)

SR-31747 (Peripheral sigma receptor antagonist)

SSR97225

STA-1474 (Prodrug of ganetespib) (HSP90 inhibitor)

Stannsoporfin (heme oxygenase inhibitor)

Streptozocin

SU14813

Sufentanil (ARX-02)

Sulforaphane (natural antioxidant)

Sunitinib

SYM-004 (anti-EGFR monoclonal antibody mixture)

SYP-0704A

Tacrolimus

TAE684 (NVP-TAE684) (ALK Inhibitor)

TAK-285 (HER2/EGFR dual kinase inhibitor)

TAK-441 (Hedghog inhibitor)

TAK-448

TAK-593 (VEGFR/PDGFR dual kinase inhibitor)

TAK-683

TAK-701 (anti-HGF monoclonal antibody)

TAK-733 (MEK inhibitor)

TAK-901 (Aurora B kinase inhibitor )

TAK-960 (PLK1 inhibitor)

Talabostat

Talampanel (AMPA-receptor antagonist)

Talaporfin sodium

Talaporfin sodium (PDT photosensitizer)

Talotrexin Ammonium

Taltobulin (tubulin inhibitor)

Tamibarotene

Tamibarotene (retinoic acid receptor (RAR) alpha/beta agonist)

Tamoxifen Citrate

Tandutinib (MLN0518) (tyrosine kinase inhibitor)

Tanomastat (matrix metalloprotease inhibitor)

Tapentadol

Tarenflurbil ((NSAID drug, enantiomer of flurbiprofen)

Tariquidar (p-glycoprotein inhibitor)

TAS-102

TAS-103 (BMS-247615)

TAS-108 (estrogenic receptor alpha (ERa) inhibitor)

TAS-109 (DNA polymerase inhibitor)

TAS266 (tetrameric Nanobody® agonist)

Tasidotin

Tasisulam (LY573636)

Tasquinimod (ABR-215050) (angiogenic inhibitor)

Tegafur

Teglarinad chloride (GMX-1777)

Telaprevir (VX-950)

Telatinib ( Tanespimycin) (Hsp90 inhibitor)

Telcagepant

Telicoplanin

Temoporfin

Temoporfin (PDT photosensitizer)

Temozolomide

Temsirolimus

Teniposide

Terameprocol (transcriptional inhibitor)

TG-0054 (CXCR4 antagonist)

TG02 (multi-kinase inhibitor of CDKs, JAK2 and FLT3)

TG100-115 (PI3K inhibitor)

TG101348 ( JAK2 inhibitor)

TGX-221 (PI3K inhibitor)

TH-302 (hypoxia-activated prodrug)

Thymectacin (NB-1011).

Ticagrelor

Tigapotide

Tigecycline

Timcodar (VX-853)

Tipifarnib (farnesyl transferase inhibitor)

Tipranavir

Tirapazamine (hypoxia toic agent)

Tivantinib (ARQ-197) (c-Met inhibitor)

Tivozanib (AV-951) (VEGFR inhibitor)

TL-310 (a taxane)

TL32711 (Smac mimetic)

Toceranib (SU11654) (Hsp90 inhibitor)

Tofacitinib (CP-690550) (JAK inhibitor)

Topotecan Hydrochloride

Tozasertib (MK-0457; VX-680) (Aurora inhibitor)

TPI-287 (ARC-100)

TPT-260

Trabectedin

Trametinib (GSK-1120212, JTP-74057) (MEK 1/2 inhibitor)

TRC093 (a humanized IgG1 monoclonal antibody)

TRC105 (human chimeric monoclonal antibody )

Treosulfan

Tretazicar (DNA alkylating agent)

Tretinoin

Triapine (ribonucleotide reductase inhibitor)

Triciribine (VQD-002) (Akt inhibitor)

TRX-518 (fully humanized IgG1 anti-huGITR Mab)

TST-88 (also see TST-10088, a recombinant protein prodrug based on a plant-derived toxin called ricin)

TSU-68

Tubacin (HDAC6 inhibitor)

Tubastatin-A (HDAC6 inhibitor)

TV-1001 (Custiren, OCX-011) [a mixed-backbone antisense oligodeoxynucleotide with chemosensitizing properties.]

TXA127 (heptapeptide COX-2 inhibitor)

U0126 (MEK inhibitor; MAP kinase inhibitor)

U3-1565 (anti-HBEGF monoclonal antibody)

Ukrain

UNBS-5162

Uracil

Uramustine (Uracil Mustard)

Uridine triacetate

Ursodeoxycholic acid ( Ursodiol)

Ursodiol ( Ursodeoxycholic acid)

V503 (human papillomavirus vaccine)

V935 (hTERT vaccine)

Vadimezan (AS-404; DMXAA) (vascular disrupting agent)

Valrubicin

Valspodar

Vandetanib (approved in 2011)

Vandetanib (approved in 2011) (VEGFR and EGFR inhibitor)

Vargatef

Varlitinib ( ARRY-543)

Vatalanib (VEGFR inhibitor)

VEL-0230 (NC-2300)

Veliparib ( ABT-888) (PARP inhibitor)

Vemurafenib

Vemurafenib (RG7204, PLX4032, RO5185426) (B-Raf inhibitor)

Verteporfin

Verteporfin (PDT photosensitizer)

Virulizin (A natural biological response modifier (BRM) isolated from bovine reticuloendothelial tissue).

Vismodegib (RG3616, GDC-0449) (Hedgehog antagonist)

Volasertib ( BI-6727) (Plk1 inhibitor)

Voreloxin (SNS-595, Vosaroxin)

Vorinostat

Vosaroxin (Voreloxin, SNS-595)

VP-701 (not available)

VTX-2337

VX-222

VX-689 (MK-5108)

VX-702 (p38 MAPK Inhibitor)

VX-745

VX-765 (Caspase inhibitor)

VX-770

WK-X-34 (P-glycoprotein inhibitors)

WYE-354 (mTOR inhibitor)

WZ4002 (EGFR inhibitor)

X-82

Xaliproden

Xen-2174 (conopeptide analog)

XL019 (JAK2 Inhibitor)

XL139 (BMS-833923)

XL147 (SAR-245408) (PI3K inhibitor)

XL228

XL281 ( BMS-908662)

XL647 (EGFR and ErbB2 inhibitor)

XL765 (SAR-245409) (PI3K/mTOR inhibitor)

XL888 (Hsp90 inhibitor)

XL999 (Spectrum Selective Kinase Inhibitor)

XMT-1001

XMT-1107

XR9051 (P-glycoprotein inhibitors)

YM-155 (Survivin inhibitor)

Zibotentan (AZD-4054, ZD4054)

ZM447439

Zoledronic Acid

Zosuquidar (P-glycoprotein inhibitor)

ZSTK474 (PI3K inhbitor)

ZYC-300 (A plasmid DNA)