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MedKoo's Collection:

 

New anticancer agents under worldwide clinical trials

 

(last update: November 30, 2011)

 

 

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Cat#      ||  Product name

201830  ||  2-methoxyestradiol (angiogenesis inhibitor)

200880  ||  4-demethylpenclomedine(also see: DMPEN) (alkylation agent)

201804  ||  AB1010 (also see: Masitinib) (tyrosine kinase inhibitor)

202170  ||  Abexinostat(also see: PCI-24781 CRA-024781) (HDAC inhibitor)

204110  ||  ABI-008 (nab-docetaxel)

204120  ||  ABI-009 (nab-rapamycin)

204130  ||  ABI-101 (nab-17AAG)

100011  ||  Abiraterone (androgen biosynthesis inhibitor)

200030  ||  Abiraterone acetate (androgen biosynthesis inhibitor)

202852  ||  ABR-215050 (also see: Tasquinimod) (angiogenic inhibitor)

201970  ||  ABT-263 (also see: Novitoclax) (Bcl-2 Inhibitor)

204140  ||  ABT-348 (temporally not available)

200040  ||  ABT-518

200044  ||  ABT-737 (BCL-2 inhibitor)

200050  ||  ABT-751

204150  ||  ABT-806 (anti-EGFR monoclonal antibody )

200051  ||  ABT-828 (a biologic compound that blocks angiogenesis of cancer cells)

203115  ||  ABT-888 (also see:  Veliparib) (PARP inhibitor)

200072  ||  AC220 (also see: Quizartinib) (FLT3 inhibitor)

200078  ||  AC480 (also see: BMS-599626) (HER inhibitor)

200079  ||  Acadesine

204160  ||  ACE-041 (an investigational protein therapeutic that inhibits angiogenesis)

204170  ||  Acolbifene

201823  ||  Acyline (also see: MER104)

204180  ||  AD-1001

200080  ||  Aderbasib (also see: INCB7839)

204190  ||  ADI-PEG20 (arginine deiminase (ADI) formulated with polyethylene glycol)

200090  ||  ADPM06

202042  ||  ADW742 (also see: NVP-ADW742)

204200  ||  AE-37 (Vaccine)

200100  ||  AEE788 (EGFR, ErbB2, KDR, and Flt-1 inhibitor)

201475  ||  AEG-40826 (also see: HGS-1029)

200110  ||  AEG-41174

204210  ||  AEW-541

202043  ||  AEW541 (also see: NVP-AEW541)

204220  ||  AEZS-108 (also see: AN-152)

200115  ||  AEZS-112 (also see: ZEN012)

200500  ||  Afatinib (also see: BIBW-2992 ) (EGFR inhibitor)

200120  ||  Afimoxifene

204230  ||  AFM-13 (a bispecific, tetravalent human antibody for Hodgkin Lymphoma.)

200123  ||  AFP-464

204240  ||  AFX-9901

204250  ||  AG-013 (Trefoil Factor)

200124  ||  AG-14699 (also see: Rucaparib, PF-01367338) (PARP1 inhibitor)

200125  ||  AG-24322

200121  ||  AG-490 (EGFR and JAK inhibitor)

204260  ||  AI-850

200127  ||  AKR-501

200130  ||  Alanosine

200131  ||  ALB-109564

200133  ||  Alendronate sodium

201931  ||  Alisertib (also see: MLN-8237) (Aurora A kinase inhibitor)

204270  ||  ALN-VSP (an RNAi therapeutic for the treatment of liver cancers )

200160  ||  ALS357 ( also see:  Betulinic acid)

204280  ||  ALT-801 (IL-2 recombinant fusion protein)

200170  ||  Alvespimycin (Hsp90 inhibitor)

200180  ||  Alvocidib (also see: Flavopiridol) (CDK inhibitor)

200182  ||  Ametantrone

200185  ||  AMG-208

204310  ||  AMG-319 (PI3 Kinase inhibitor  )

204320  ||  AMG-337 (c-Met inhibitor)

204330  ||  AMG-386 (angiopoietin inhibitor, an anti-angiopoietin peptibody)

201934  ||  AMG-706 (also see: Motesanib ) (tyrosine kinase inhibitor)

204340  ||  AMG-780 (anti-angiopoietin antibody )

204350  ||  AMG-820 (antibody that targets c-fms and decreases tumor TAM function)

204360  ||  AMG-888 (antibody that inhibits HER3 oncogenic signaling)

204370  ||  AMG-900 (inhibitor of Aurora kinases A, B, and C.)

200200  ||  Amonafide dihydrohloride

200210  ||  Amonafide malate (also see: AS-1413)

200220  ||  Amrubicin

200720  ||  Amsilarotene (also see: TAC-101)

201950  ||  Amuvatinib (also see: MP-470)

204220  ||  AN-152 (also see: AEZS-108)

204371  ||  AN-207

200252  ||  AN-2728 (PDE4 inhibitor)

200257  ||  ANA-773

200230  ||  Anamorelin hydrochloride

205475  ||  ANG-1005 (also see: GRN-1005)

200240  ||  Annamycin

200250  ||  ANX-510

204380  ||  ANX-514 (docetaxel new formulation)

200255  ||  ANZ-207 (cancer vaccine)

202320  ||  AP-24534 (also see: Ponatinib) (tyrosine kinase inhibitor)

200135  ||  Apatinib (VEGFR inhibitor)

200140  ||  Apaziquone (bioreductive prodrug, hypoxia toxic agent)

200150  ||  Aplidine (also see: Plitidepsin)

205484  ||  APN01 (also See: GSK-2586881)

200270  ||  APO-866 (also See: FK866) (NAMPT inhibitor)

200273  ||  Apricoxib

200272  ||  AR-12 (also see: OSU-03012)

200275  ||  AR-42

200274  ||  AR-67(also see: Silatecan , also see: DB-67)

202964  ||  ARC-100 ( also see: TPI-287)

204420  ||  ARN-509 (androgen receptor antagonist)

200280  ||  Aroplatin

200281  ||  ARQ-092 (AKT inhibitor)

200283  ||  ARQ-197 (also see: Tivantinib) (c-Met inhibitor)

200284  ||  ARQ-501 (also see:  R1668,  beta-lapachone)

204430  ||  ARQ-621

204440  ||  ARQ-736 (BRAF Inhibitor)

205531  ||  ARRY-162 (also see: MEK-162) (MEK1/2  inhibitor)

200290  ||  ARRY-300 (MEK inhibitor)

200291  ||  ARRY-380

200292  ||  ARRY-520

205660  ||  ARRY-543 ( also see: Varlitinib)

200294  ||  ARRY-614

200313  ||  ARRY-704 (also see: AZD-8330 )

205633  ||  ARX-02 (also see: Sufentanil)

200310  ||  Arzoxifene

200210  ||  AS-1413 (also see: Amonafide malate)

200296  ||  AS-605240

200297  ||  AS-703026 (MEK ½ inhibitor)

202422  ||  AS703569(also see: R763 )

204450  ||  ASP-3026

200314  ||  AT-101(also see: Gossypol acetic acid)

200317  ||  AT-13387

204460  ||  AT-406

200320  ||  AT-7519

200322  ||  AT-9283 (multikinase inhibitor)

200330  ||  Atamestane

200340  ||  Atiprimod

200350  ||  ATN-161

200360  ||  ATN-224

200370  ||  Atrasentan

200371  ||  AUY-922 (also see: NVP-AUY922,  VER-52296) (Hsp90 inhibitor)

201944  ||  AV-412 (also see: MP-412)  (EGFR/HER2 tyrosine kinase inhibitor)

202955  ||  AV-951 (also see: Tivozanib) (VEGFR inhibitor)

200380  ||  AVE8062(also see: Ombrabulin )

204480  ||  AVL-292

200390  ||  AVN-944 (also see: VX-944) (IMPDH inhibitor)

200400  ||  Axitinib (VEGFR inhibitor)

200410  ||  AZD-0530 (also see: Saracatinib) (Src and Abl inhibitor)

200420  ||  AZD-1152 (also see: Barasertib) (Aurora B inhibitor)

200421  ||  AZD1152-HQPA (Aurora B inhibitor)

204510  ||  AZD-1480 (JAK2 inhibitor)

204520  ||  AZD-2014

200423  ||  AZD-2281 (also see: Olaparib) (PARP inhibitor)

204530  ||  AZD-2461

204540  ||  AZD-3514

203200  ||  AZD-4054 (also see: Zibotentan,  ZD4054)

204550  ||  AZD-4547 (pan-FGFR inhibitor)

200422  ||  AZD-4769

200424  ||  AZD-4877

200425  ||  AZD-4992

205669  ||  AZD-5363 (PKB/Akt inhibitor)

200426  ||  AZD-5438 (CDK Inhibitor)

200427  ||  AZD-6126

200300  ||  AZD-6244 (also see: Selumetinib) (MEK 1/2 inhibitor)

200310  ||  AZD-6918

200311  ||  AZD-7762 (checkpoint kinase inhibitor)

200312  ||  AZD-8055 (mTOR inhibitor)

200313  ||  AZD-8330 (also see: ARRY-704)

200298  ||  AZD-8931 (HER1and HER2 inhibitor)

200315  ||  AZM-475271

200316  ||  Bafetinib (also see: INNO-406)

200430  ||  Banoxantrone (hypoxia toxic agent)

200420  ||  Barasertib (also see: AZD-1152) (Aurora B inhibitor)

202530  ||  Bardoxolone methyl (also see: RTA402)

200440  ||  Batabulin sodium

200442  ||  Batimastat

204560  ||  BAY 10-00394

202436  ||  BAY 73-4506 (also see: Regorafenib) (oral multi-kinase inhibitor)

204610  ||  BAY 79-4620 (Antibody–drug conjugate)

204570  ||  BAY 80-6946

204590  ||  BAY 94-9392

202431  ||  BAY86-9766 (also see: RDEA119) (MEK inhibitor)

201802  ||  BB-2516 (also see: Marimastat)

204620  ||  BBI-608

204630  ||  BC-819 (a plasmid comprised of the H19 gene regulatory sequences )

200450  ||  Becatecarin

200455  ||  Beclometasone dipropionate

200460  ||  Belinostat (HDAC inhibitor)

200461  ||  Belotecan

200470  ||  Bendamustine HCl

200480  ||  Beraprost

200490  ||  Berubicin

200284  ||  beta-lapachone (also see:  R1668,  ARQ-501)

200160  ||  Betulinic acid ( also see:  ALS357)

204920  ||  Bevonium methylsulfate (also see CG-201)

200491  ||  BEZ235 ( also see: NVP-BEZ235)

204790  ||  Bezielle (also see: BZL-101)

204790  ||  Bezielle (also see:  BZL-101)

202270  ||  BGC-9331 (also see: Plevitrexed)

209490  ||  BGC-945 (also see: ONX-0801)

204640  ||  BGJ-398 (pan FGFR kinase inhibitor)

200492  ||  BGT-226

204650  ||  BHQ-880 (Antibody)

200493  ||  BI-2536 (Polo-like kinase 1 inhibitor)

204660  ||  BI-505 (anti-ICAM-1 monoclonal antibody BI-505 )

200494  ||  BI-6727 (also see: Volasertib) (Plk1 inhibitor)

204670  ||  BI-811283

200495  ||  BI-831266 (Not available temporially)

200496  ||  BIBF-1120 (also see: Intedanib ) (VEGFR inhibitor)

200500  ||  BIBW-2992 (also see: Afatinib) (EGFR inhibitor)

204665  ||  BIIB-015 (DM4-conjugated anti-Cripto monoclonal antibody )

200505  ||  BIIB-021 (also see: CNF2024) (HSP90 inhibitor)

204670  ||  BIIB-022 (a human, nonglycosylated IgG4 monoclonal antibody)

204680  ||  BIW-8962 (anti-ganglioside GM2 monoclonal antibod)

200515  ||  BIX-02188

204690  ||  BKM-120 (PI3K inhibitor)

204710  ||  BMN-673

202834  ||  BMS-247615 (also see: TAS-103)

200520  ||  BMS-275183

202640  ||  BMS-387032 (also see: SNS-032)

200521  ||  BMS-536924

200524  ||  BMS-536924

200078  ||  BMS-599626 (also see: AC480) (HER inhibitor)

200531  ||  BMS-641988

200533  ||  BMS-690514

201275  ||  BMS-753493(also see: Epofolate )

200534  ||  BMS-754807 (IGF-1R inhibitor)

200527  ||  BMS-777607 (Met tyrosine kinase inhibitor)

200535  ||  BMS-833923 (also see: XL-139)

204730  ||  BMS-908662 (also see: XL281)

204740  ||  BMS-936558 (an anti-programmed death-1 (MDX-1106))

204750  ||  BMS-936559 (an anti-programmed death-1)

200540  ||  BN2629 (also see: SJG-136, SG2000)

200550  ||  BN83495 (also see: STX64, Irosustat)

204760  ||  BNC-105

201630  ||  BNP-1350 (also see: Cositecan, Karenitecin )

200560  ||  Bosutinib (Abl and Src  inhibitor)

200561  ||  BQS-481

200569  ||  Brivanib (VEGFR2 inhibitor)

200570  ||  Brivanib alaninate (VEGFR2 inhibitor)

202520  ||  Brivudin (also see: RP-101)

200580  ||  Brostallicin

200582  ||  BSI-201 (also see: Iniparib) (PARP inhibitor)

204770  ||  BT-062 (Anti-myeloma monoclonal antibody-DM4 immunoconjugate)

200584  ||  BTZ043

204780  ||  BYL-719

204790  ||  BZL-101 (also see: Bezielle)

204810  ||  C31510 (not available)

200800  ||  CA4P (also see: combretastatinA-4phosphate, Fosbretabulin)

200585  ||  Cabazitaxel (also see: XRP-6258)

200595  ||  Cabozantinib (also see:  XL-184) (VEGFR2, Met, FLT3, Tie2, Kit and Ret inhibitor)

200586  ||  CAL-101 (PI3K inhibitor)

204820  ||  CALAA-01 (siRNA-based cancer drug)

200590  ||  Calcitriol

200600  ||  Canertinib

200610  ||  Canfosfamide

201453  ||  Capesaris (Also see: GTX-758)

200620  ||  Carbendazim

204830  ||  Carboxyamidotriazole orotate  (CTO)

200630  ||  Carfilzomib (proteasome inhibitor)

200650  ||  Casopitant mesylate

202600  ||  CB1089 (also see: Seocalcitol)

204840  ||  CB-1400 (Not Available)

202020  ||  CB-3304 (also see: Noscapine)

202385  ||  CBLC102 (also see: Quinacrine; Mepacrine)

204860  ||  CBP-501

204870  ||  CC-223

200651  ||  CC-401

200670  ||  CC-8490

200680  ||  CDB-4124

204880  ||  CDX-011 (antibody-drug conjugate).

204890  ||  CDX-1401 (fusion protein / antibody )

200690  ||  Cediranib dihydrochloride

200694  ||  Celastrol (HSP90 inhibitor)

200700  ||  Celecoxib

200710  ||  Cemadotin

200712  ||  CEP-11981

200713  ||  CEP-18770

200716  ||  CEP-7055

204910  ||  CEP-9722

200721  ||  Cerovive (also see: NXY-059)

200730  ||  Cevipabulin (antimicrotubule agent)

200740  ||  CF-101

204920  ||  CG-201 (also see Bevonium methylsulfate)

200750  ||  CGC-11047 (also see: PG-11047)

200752  ||  CGS-21680 (adenosine A2A receptor agonist)

200755  ||  Chelerythrine chloride

204930  ||  Chidamide  (also see: CS055HBI-8000)

200760  ||  CHIR258 (also see: TKI-258, Dovitinib)

200770  ||  CHIR-265 (also  see: RAF-265)

200774  ||  CHIR-99021

200776  ||  CHS-828 (NAD inhibitor)

200771  ||  CI-1040 (also  see: PD184352)

200780  ||  Cilengitide

200781  ||  CJ-15161

205612  ||  CKI27 (also see: RG7304)

200790  ||  Clodronate disodium

204940  ||  CLR-1404

204950  ||  CLT-008 (human myeloid progenitor cells)

200791  ||  CNDO-101

200505  ||  CNF2024 (also see: BIIB-021) (HSP90 inhibitor)

204960  ||  CNTO-95 (a fully human monoclonal IgG1 antibody)

204970  ||  CO-101 (also  see: CP-4126) (antimetabolite agent)

200800  ||  CombretastatinA-4phosphate(also see: Fosbretabulin , CA4P)

200793  ||  Cordycepin (also  see: OVI-123)

201630  ||  Cositecan (also see: BNP-1350, Karenitecin ).

204970  ||  CP-4126 (also  see: CO-101) (antimetabolite agent)

200810  ||  CP-547632

200811  ||  CP-690550

200820  ||  CP-724714

205020  ||  CP-868596 (also see: Crenolanib )

200823  ||  CPI-613

205260  ||  CPP-1X (also see: Eflornithine)

204990  ||  CPX-1

205010  ||  CPX-351

202170  ||  CRA-024781(also see: Abexinostat PCI-24781) (HDAC inhibitor)

205020  ||  Crenolanib (also see: CP-868596)

202222  ||  Crizotinib (also see: PF-2341066) (tyrosine kinase inhibitor)

205030  ||  CRLX-101

200831  ||  Crolibulin (also see: EPC2407)

205050  ||  CRS-100 [a live-attenuated strain of Listeria monocytogenes (Lm)]

205060  ||  CRS-207 [a weakened (attenuated) form of Listeria monocytogenes]

204930  ||  CS055  (also see ChidamideHBI-8000)

205250  ||  CS-7017 (also see: Efatutazone, inolitazone)

205070  ||  CST-101 (the native NK-92 cell-line)

205080  ||  CT-011 (a humanized monoclonal antibody (mAb) that modulates the immune response and inhibits tumor growth and the spread of metastases.)

200841  ||  CUDC-101 (HDAC, EGFR and HER2 inhibitor)

205090  ||  Custiren (also see: TV-1001, also see: OCX-011) [a mixed-backbone antisense oligodeoxynucleotide with chemosensitizing properties.]

205110  ||  CV9103 (mRNA-derived prostate cancer vaccine)

200842  ||  CVT-6883 (A2B adenosine antagonist)

202380  ||  CX-3543 (also see: Quarfloxin)

200843  ||  CX-4945

200848  ||  CX-5461

200844  ||  CYC-116 (Aurora kinase/VEGFR2 inhibitor)

205130  ||  CYT-107 (Interleukin-7)

200786  ||  CYT-387 (JAK inhibitor)

205140  ||  CYT-6091 (a nanotherapeutic manufactured by covalently linking tumor necrosis factor-a (TNF) onto the surface of 30 nm particles of pegylated colloidal gold)

205653  ||  D-3263

205479  ||  Dabrafenib (Also see: GSK-2118436) (B-RAF inhibitor)

200845  ||  Dacinostat (also see: NVP-LAQ824)

205576  ||  Dacomitinib (also see: PF-00299804) (EGFR inhibitor)

200846  ||  Danusertib

200850  ||  Darinaparsin (also see: ZIO-101)

200274  ||  DB-67 (also see: AR-67, also see: Silatecan)

200851  ||  DCC-2036

200860  ||  Deforolimus (also see: Ridaforolimus)

100255  ||  Degarelix acetate

200890  ||  Denibulin (also see: MN-029)

201000  ||  Dexmethylphenidate hydrochloride

200900  ||  Diethylnorspermine

201020  ||  Diflomotecan

201030  ||  Dimesna

202572  ||  Dinaciclib (also see: SCH-727965, PS-095760) (CDK inhibitor)

202881  ||  DJ-927 (also see: Tesetaxel )

200880  ||  DMPEN(also see: 4-demethylpenclomedine) (alkylation agent)

201050  ||  DMXAA(also see: Vadimezan )

201060  ||  Docosahexaenoic acid

201065  ||  Dofequidar

201040  ||  Doramapimod

200760  ||  Dovitinib (also see: TKI-258,  CHIR258)

201070  ||  Dutasteride

201071  ||  E6201

205150  ||  E7016

201072  ||  E7050

201080  ||  E7080 (also see: lenvatinib)

205160  ||  E7272 (also see : ONTAK or denileukin diftitox)

201290  ||  E7389 (also see: Eribulin mesylate )

201090  ||  E7820

201100  ||  E7974

205170  ||  EC-0225

205180  ||  EC-0489

205190  ||  EC-145

205210  ||  EC-17

205230  ||  EC-20

205240  ||  ECC-33 (also see: RG7686) [monoclonal antibody]

201150  ||  Edatrexate

201160  ||  Edotecarin

201180  ||  Efaproxiral

205250  ||  Efatutazone (also see: CS-7017, inolitazone)

205260  ||  Eflornithine (also see: CPP-1X)

205270  ||  EGEN-001 [non-viral vector consisting of a plasmid DNA encoding the human gene for interleukin 12 (IL-12)]

205280  ||  EGEN-002 [not available]

202190  ||  EKB569 (also see: Pelitinib) (pan-ErbB tyrosine kinase inhibitor )

201190  ||  Elacridar

201195  ||  Elacytarabine (antimetabolite agent)

201200  ||  Elagolix (also see:  NBI-56418)

201210  ||  Elesclomol (HSP-90 Inhibitor)

201220  ||  Elinafide

202300  ||  Elisidepsin (also see: PM-02734)

201230  ||  Elsamitrucin

201240  ||  Eltrombopag

205492  ||  EMD1201081 (also see: IMO-2055)

205330  ||  EMD-1204831

201245  ||  EMD-1214063 (c-Met inhibitor)

201250  ||  Eniluracil

201260  ||  ENMD-1198

201264  ||  ENMD-2076 (Aurora kinase inhibitor)

201266  ||  Entinostat (also see: MS-275,  SNDX-275) (HDAC inhibitor)

201270  ||  Enzastaurin (also see: LY317615)

205340  ||  EP-100 [an LHRH receptor-targeting ligand conjugated to a novel
membrane-disrupting peptide called CLIP 71.]

200831  ||  EPC2407 (also see: Crolibulin)

202160  ||  EPO906 (also see: Patupilone)

201275  ||  Epofolate (also see: BMS-753493)

201280  ||  Epothilone D

201290  ||  Eribulin mesylate (also see: E7389)

205510  ||  Erismodegib (also see: LDE225, NVP-LDE225) (Smo antagonist)

201300  ||  ES285

201310  ||  Etalocib

205350  ||  ETBX-011 (an immunotherapeutic to treat colorectal cancer)

201320  ||  Ethonafide

201330  ||  Ethynylcytidine

100335  ||  Everolimus

201340  ||  Exatecan

201372  ||  EXEL-2880 (also see: XL888, SK1363089, GSK089, Foretinib ) (MET/VEGFR2 inhibitor)

201350  ||  Exherin

201354  ||  Exisulind

201360  ||  Ezatiostat hydrochloride

205380  ||  EZN-2208 (Pegylated SN-38)

205410  ||  EZN-2968 [a novel hypoxia-inducible factor-1a messenger ribonucleic acid antagonist (IC50 ~1-5 nM)]

205420  ||  EZN-3042 [a locked nucleic acid antisense oligonucleotide].

205430  ||  Fenretinide

205440  ||  FG-3019 (anti-CTGF monoclonal antibody)

205450  ||  Finasteride

200270  ||  FK866 (also See: APO-866) (NAMPT inhibitor)

200180  ||  Flavopiridol (also see: Alvocidib) (CDK inhibitor)

205460  ||  Fluciclatide F-18

201380  ||  Fludarabine

201372  ||  Foretinib (also see: XL888, SK1363089, GSK089, EXEL-2880) (MET/VEGFR2 inhibitor)

201390  ||  Forodesine

205461  ||  Fosaprepitant

200800  ||  Fosbretabulin (also see: combretastatinA-4phosphate, CA4P)

201393  ||  Fostamatinib

205588  ||  FP-1039 (A soluble fusion protein)

205463  ||  FP-1039 (an FGFR1-Fc fusion protein)

205465  ||  FT-1050

205646  ||  Galeterone (also see: TOK-001)

202703  ||  Ganetespib (also see: STA-9090)

205467  ||  GDC-0068 (AKT  inhibitor)

203500  ||  GDC-0449 (also see: RG3616, Vismodegib) (Hedgehog antagonist)

205468  ||  GDC-0917

201395  ||  GDC-0941 (PI3K inhibitor)

203185  ||  GDC-0973 (also see: XL518) (MEK inhibitor)

205470  ||  GDC-0980 (also see: RG7422) ( PI3 kinase/mTOR inhibitor)

205471  ||  GENZ-644282

205472  ||  GGTI-2418

205473  ||  GI-4000 (Targeted Molecular Immunogen)

205474  ||  GI-6207 (vaccine)

201410  ||  Gimatecan

201420  ||  Glufosfamide

202860  ||  GMX-1777 (also see: Teglarinad chloride) 

201422  ||  Golotimod

201430  ||  Gossypol

200314  ||  Gossypol acetic acid (also see: AT-101)

201436  ||  GPI-15427

201440  ||  GPX100

201450  ||  GPX150

205475  ||  GRN-1005 (also see: ANG-1005)

205489  ||  GRN-163L (also see: Imetelstat)

205476  ||  GS-6624  (humanized monoclonal antibody)

205569  ||  GS7904L (also  see: OVI-237, OSI-7904L)

201452  ||  GS-9219

201372  ||  GSK089 (also see: XL888, SK1363089, Foretinib, EXEL-2880) (MET/VEGFR2 inhibitor)

201456  ||  GSK1070916

205477  ||  GSK-1070916A

201458  ||  GSK-1120212 (aslo see: Trametinib, JTP-74057) (MEK 1/2 inhibitor)

205478  ||  GSK-2110183 (Akt inhibitor)

205479  ||  GSK-2118436 (Also see: Dabrafenib) (B-RAF inhibitor)

205480  ||  GSK-2126458 (PI3K inhibitor)

205481  ||  GSK-2141795 (Akt inhibitor)

205482  ||  GSK-2256098

205483  ||  GSK-2401502

205484  ||  GSK-2586881 (also See: APN01)

205667  ||  GSK-461364  (PLK Inhibitor)

205670  ||  GSK-690693 (pan-Akt kinase inhibitor)

201453  ||  GTX-758 (Also see: Capesaris)

202161  ||  GW786034 (also see: Pazopanib Hydrochloride) (tyrosine kinase inhibitor )

202050  ||  GX15-070 (also see: Obatoclax  )

201460  ||  HA14-1

204930  ||  HBI-8000  (also see: CS055Chidamide)

205485  ||  HE-3235

201466  ||  Hesperadin

201475  ||  HGS-1029 (also see: AEG-40826)

201470  ||  HKI272 (also see: Neratinib) (HER2 and EGFR inhibitor)

201480  ||  HMN-176

201490  ||  HMN-214

202075  ||  Homoharringtonine(also see: Omacetaxine mepesuccinate )

205486  ||  HQK-1004

201491  ||  HRC-302 (Hemosol cell therapy)

205487  ||  HSP-990

201495  ||  Hypothemycin

205488  ||  Iboctadekin  (immunostimulatory cytokine )

201684  ||  Ibutamoren

205489  ||  Imetelstat  (also see: GRN-163L)

201500  ||  Imexon

205490  ||  IMGN-388 (Targeted Antibody Payload, TAP)

205491  ||  IMGN-901 (lorvotuzumab mertansine)

201510  ||  Imidazoacridone

205492  ||  IMO-2055 (also see: EMD1201081)

201512  ||  INCB-18424 (also see: Ruxolitinib) (JAK1 inhibitor)

205493  ||  INCB-24360

205494  ||  INCB-28060

200080  ||  INCB7839 (also see: Aderbasib)

201520  ||  Incyclinide

201530  ||  Indibulin (also see: ZIO-301)

201540  ||  Indisulam

201545  ||  Ingenol Mebutate (also see: PEP005)

200582  ||  Iniparib (also see: BSI-201) (PARP inhibitor)

205495  ||  INK-128 (mTOR inhibitor)

201550  ||  INNO-206 (DNA intercalating agent)

200316  ||  INNO-406 (also see: Bafetinib)

201561  ||  INO-1001

205250  ||  Inolitazone(also see: CS-7017, Efatutazone )

201562  ||  INSM-18

200496  ||  Intedanib (also see:  BIBF-1120)  (VEGFR inhibitor)

201570  ||  Iobenguane

205496  ||  Ioflubenzamide I-131 (also see: MIP-1145)

205497  ||  IPH-2101 (human anti-NK-cell inhibitory receptor mAb)

201571  ||  IPI-493

202450  ||  IPI504 (also see: Retaspimycin) (HSP90 inhibitor)

201572  ||  IPI-926

201580  ||  Irofulven

200550  ||  Irosustat (also see: STX64, BN83495)

201590  ||  Isatoribine

205499  ||  ISF-35 (vaccine)

202000  ||  isocoumarin (also see: NM-3)

201600  ||  Ispinesib

201610  ||  Ixabepilone

201611  ||  JI-101

201612  ||  JNJ-26481585

201613  ||  JNJ-26483327

201614  ||  JNJ-26854165 (also see: Serdemetan)

201615  ||  JNJ-38877605 (tyrosine kinase inhibitor)

201458  ||  JTP-74057 (aslo see: Trametinib, GSK-1120212) (MEK 1/2 inhibitor)

205502  ||  JX-594 (thymidine kinase-deleted vaccinia-hGM-CSF)

205503  ||  JX-929 (A highly tumor-selective vaccinia virus )

201620  ||  Kahalalide F

201630  ||  Karenitecin (also see: CositecanBNP-1350).

205504  ||  KB-004 (Humaneered™ monoclonal antibody)

201640  ||  Ketamine

205505  ||  KHK-2866 (Anti-HB-EGF Antibody)

201650  ||  KOS-1584 (also see: R1645)

201660  ||  KRN5500

201670  ||  KRX-0402

203060  ||  KRX-0601(also  see UCN-01)

201681  ||  KU-55933

201684  ||  KW-2449

205506  ||  KW-2478 (Hsp90 inhibitor)

201686  ||  KX2-391

205508  ||  Lansoprazole

201705  ||  Laromustine(also see: VNP40101M)

201710  ||  Larotaxel (also see: XRP9881)

201720  ||  Lasofoxifene

202151  ||  LBH589 (also see: Panobinostat; NVP-LBH589) (HDAC inhibitor)

205509  ||  LCL-161

205510  ||  LDE225 (also see: Erismodegib, NVP-LDE225) (Smo antagonist)

205511  ||  LDK-378

205512  ||  LE-DT (Liposome Encapsulated Docetaxel)

205513  ||  LEE-011

201724  ||  Lemuteporfin (also see: QLT-0074)

201080  ||  lenvatinib (also see: E7080)

205514  ||  LEP-ETU (liposomal paclitaxel, also see: PNU-93914)

205515  ||  LEQ-506

201730  ||  Lestaurtinib

100542  ||  Levoleucovorin Calcium

201741  ||  LGD-4665

200060  ||  Linifanib ( also see: ABT869)

202096  ||  Linsitnib (also see: OSI-906) (IGF-1R inhibitor)

205521  ||  Litronesib (aslo see: LY2523355)

201750  ||  Lomeguatrib

201760  ||  Lonafarnib

205517  ||  LOR253

201761  ||  LP-261

201780  ||  Lucanthone

205518  ||  LY2090314

205520  ||  LY2157299 (type I receptor TGF-beta kinase antagonist)

205519  ||  LY2181308 (antisense oligonucleotide)

201792  ||  LY2334737 (antimetabolite agent)

205521  ||  LY2523355 (aslo see: Litronesib)

205522  ||  LY2584702

201794  ||  LY2603618

205523  ||  LY2606368

205524  ||  LY2624587 (not available)

205525  ||  LY2780301 (AKT inhibitor)

205526  ||  LY2801653

205527  ||  LY2874455

205528  ||  LY2875358 (anti-c-MET monoclonal antibody)

201795  ||  LY294002 (PI3K inhibitor)

205529  ||  LY2940680

201270  ||  LY317615 (also see: Enzastaurin)

202851  ||  LY573636 (also see: Tasisulam)

201800  ||  M40403

201802  ||  Marimastat (also see: BB-2516)

202031  ||  Marizomib (also see: NPI-0052) (proteasome inhibitor)

201804  ||  Masitinib (also see: AB1010) (tyrosine kinase inhibitor)

201810  ||  MB07133

201821  ||  MDV3100

205530  ||  Mechlorethamine Gel

205531  ||  MEK-162 (also see: ARRY-162) (MEK1/2  inhibitor)

202385  ||  Mepacrine (also see: Quinacrine; CBLC102)

201823  ||  MER104 (also see: Acyline)

203160  ||  Mesupron (also see: WX-671)

205650  ||  Methoxyamine (also see: TRC102)

205533  ||  Methyl aminolevulinate

205671  ||  MG-516 (multi-targeted kinase inhibitor)

201933  ||  MGCD-0103 (also see: Mocetinostat)  (HDAC inhibitor)

201841  ||  MGCD-265 (multitargeted tyrosine kinase inhibitor)

201850  ||  Midostaurin (also see: PKC412)

201860  ||  Mifamurtide

201870  ||  Mifepristone

201880  ||  Milataxel

201890  ||  Miltefosine

205535  ||  MINT-1526A (An anti-murine integrin α5β1 antibody)

205536  ||  MIP-1095

205496  ||  MIP-1145 (also see: Ioflubenzamide I-131)

201891  ||  MK-0429

201900  ||  MK-0457 (also  see Tozasertib VX-680)  (Aurora inhibitor)

201910  ||  MK-0731

201911  ||  MK-0752

202062  ||  MK-0822 (also see: Odanacatib)  (protease inhibitor)

205537  ||  MK-1496

201912  ||  MK-1775 (WEE inhibitor)

201913  ||  MK-2206 (Akt inhibitor)

201914  ||  MK-2461

201915  ||  MK-4101 (not available)

201916  ||  MK-4827 (PARP inhibitor)

201917  ||  MK-5108 (also see: VX-689)

201918  ||  MK-8033

201920  ||  MKC-1

205539  ||  MKC1106-PP (immunotherapy)

201922  ||  MKI-833

202790  ||  MLN0518 (also see: Tandutinib) (tyrosine kinase inhibitor)

201924  ||  MLN-4924

201930  ||  MLN-8054 (aurora kinase inhibitor)

201931  ||  MLN-8237 (also see: Alisertib) (Aurora A kinase inhibitor)

205541  ||  MLN-9708 (also see: Ixazomib)

205542  ||  MM-111 (a bispecific antibody).

205720  ||  MM-302 (doxorubicin nanotherapy)

205543  ||  MM-398 (irinotecan nanotherapy)

200890  ||  MN-029 (also see: Denibulin)

201932  ||  MN-201

201933  ||  Mocetinostat (also see: MGCD-0103) (HDAC inhibitor)

201934  ||  Motesanib (also see: AMG-706) (tyrosine kinase inhibitor)

201940  ||  Motexafin gadolinium

201942  ||  Motexafin lutetium

201944  ||  MP-412 (also see: AV-412) (EGFR/HER2 tyrosine kinase inhibitor)

201950  ||  MP-470 (also see: Amuvatinib)

201951  ||  MPC-2130

205544  ||  MPC-3100

201960  ||  MPC-6827 (also see: Verubulin)

205545  ||  MRX-1024

201266  ||  MS-275 (also see: Entinostat,  SNDX-275) (HDAC inhibitor)

201961  ||  MSX-122

205546  ||  MT-110 (a Bispecific T cell Engager (BiTE)® antibody)

205547  ||  Muparfostat  (also see: PI88, heparin sulfate)

205548  ||  MVA-5T4 (attenuated modified Vaccinia Ankara virus)

205549  ||  Nabiximols

201955  ||  NB-1011 (also see: Thymectacin).

201980  ||  NBI-42902

201200  ||  NBI-56418 (also see:  Elagolix)

203111  ||  NC-2300 (also see: VEL-0230)

201824  ||  Nemorubicin

201470  ||  Neratinib (also see: HKI272) (HER2 and EGFR inhibitor)

201985  ||  Netupitant

201990  ||  Nilotinib (Bcr-Abl inhibitor)

205551  ||  NK-012

205740  ||  NKP-1339

205742  ||  NKP-2235

205552  ||  NKTR-102

205553  ||  NKTR-105

202000  ||  NM-3 (also see: isocoumarin)

205554  ||  NMS-1116354

205555  ||  NMS-1286937

202010  ||  Nolatrexed

205556  ||  Norepinephrine

202020  ||  Noscapine (also see CB-3304)

202030  ||  NOV-002

201970  ||  Novitoclax (also see: ABT-263) (Bcl-2 Inhibitor)

202031  ||  NPI-0052 (also see: Marizomib) (proteasome inhibitor)

202040  ||  NPI-2358 (also see: Plinabulin)

202041  ||  NRX-4204

205557  ||  NTX-10 (vaccine)

205558  ||  NV-1020 (oncolytic herpes simplex virus type 1)

202042  ||  NVP-ADW742 (also see: ADW742)

202043  ||  NVP-AEW541 (also see:  AEW541)

200371  ||  NVP-AUY922 (also see: AUY-922, VER-52296) (Hsp90 inhibitor)

200491  ||  NVP-BEZ235 ( also see: BEZ235)

200845  ||  NVP-LAQ824 (also see: Dacinostat)

202151  ||  NVP-LBH589 (also see: Panobinostat; LBH589) (HDAC inhibitor)

205510  ||  NVP-LDE225 (also see: LDE225, Erismodegib) (Smo antagonist)

202045  ||  NVP-TAE684 (also see: TAE684) (ALK Inhibitor)

200721  ||  NXY-059 (also see: Cerovive)

202050  ||  Obatoclax ( also see:   GX15-070) (BCL-2 Inhibitor)

205559  ||  Oblimersen  (bcl-2 antisense oligodeoxynucleotide G3139)

205560  ||  OBP-301 (Telomerase-Specific Replication-Competent Adenovirus)

202087  ||  OC144-093 (also see: ONT-093)

205090  ||  OCX-011 (also see: Custiren, also see: TV-1001) [a mixed-backbone antisense oligodeoxynucleotide with chemosensitizing properties.]

202062  ||  Odanacatib (also see: MK-0822) (protease inhibitor)

202064  ||  Oglufanide

205561  ||  OGX-427 (Hsp27 antisense oligonucleotide )

200423  ||  Olaparib (also see: AZD-2281) (PARP inhibitor)

202070  ||  Oleandrin (also see: PBI-05204)

202075  ||  Omacetaxine mepesuccinate (also see: Homoharringtonine)

200380  ||  Ombrabulin (also see: AVE8062)

200385  ||  Omtriptolide

205563  ||  ON-013105

202080  ||  ON-01910 also see: Rigosertib)

202087  ||  ONT-093 (also see: OC144-093)

205625  ||  ONX 0805 (also see: SB1578)

209490  ||  ONX-0801 (also see: BGC-945)

205565  ||  ONX-0912

205730  ||  ONX-0914

205566  ||  OPB-31121

205567  ||  OPB-51602

202090  ||  Ortataxel

200724  ||  Orteronel (also see: TAK-700)

202094  ||  OSI-027 (mTOR inhibitor)

205569  ||  OSI-7904L(also  see: GS7904L, OVI-237 )

202096  ||  OSI-906 (also see: Linsitnib) (IGF-1R inhibitor)

202100  ||  OSI-930

202103  ||  Ostarine (also see: MK-2866, GTX-024)

202103  ||  MK-2866 (also see: Ostarine, GTX-024)

202103  ||  GTX-024 (also see: MK-2866, Ostarine)

202102  ||  OSU-03012

200272  ||  OSU-03012 (also see: AR-12)

202101  ||  OVI­123 (also  see: Cordycepin)

200793  ||  OVI-123 (also  see: Cordycepin)

205569  ||  OVI-237 (also  see: GS7904L, OSI-7904L)

205570  ||  OXi-4503

202110  ||  Ozarelix (also  see: SPI-153)

202114  ||  P2045

202118  ||  P276-00

205571  ||  PA-799 (not available)

202571  ||  Pacritinib (also see: SB1518)

202185  ||  Padoporfin   (also see: Tookad)

202130  ||  Palifosfamide (also see: ZIO-201)

202133  ||  Palomid 529 (PI3K inhibitor; Akt inhibitor; mTOR inhibitor)

202151  ||  Panobinostat (also see: NVP-LBH589; LBH589) (HDAC inhibitor)

205572  ||  Pasireotide (also see: SOM-230)

202160  ||  Patupilone (also see: EPO906)

202161  ||  Pazopanib Hydrochloride (also see: GW786034) (tyrosine kinase inhibitor )

202070  ||  PBI-05204 (also see: oleandrin)

202170  ||  PCI-24781(also see: Abexinostat CRA-024781) (HDAC inhibitor)

205574  ||  PCI-27483

202171  ||  PCI-32765 (BTK inhibitor)

202172  ||  PD-0325901 (MEK inhibitor)

202173  ||  PD-0332991 (CDK Inhibitor)

202174  ||  PD-153035 (EGFR inhibitor)  

200771  ||  PD184352 (also  see: CI-1040)

202190  ||  Pelitinib (also see: EKB569) (pan-ErbB tyrosine kinase inhibitor)

202200  ||  Pelitrexol

201545  ||  PEP-005 (also see:  Ingenol Mebutate)

202220  ||  Perifosine (AKT Inhibitor)

205576  ||  PF-00299804 (also see: Dacomitinib) (EGFR inhibitor)

202228  ||  PF-00562271 (also see: PF-562271)

200124  ||  PF-01367338 (Also see: Rucaparib, AG-014699) (PARP1 inhibitor)

202224  ||  PF-03084014

205580  ||  PF-03446962 (anti-ALK-1 monoclonal antibody)

205581  ||  PF-03758309 (PAK4 inhibitor)

205582  ||  PF-04449913

205583  ||  PF-04554878

205584  ||  PF-04605412 (anti-A5B1 integrin monoclonal antibody )

202226  ||  PF-04691502 (PI3K/mTOR inhibitor)

205586  ||  PF-04856884 (also see: CVX-060) [the fusion of two Ang2 sequestering peptides]

202255  ||  PF-05212384 (also see: PKI-587)

202222  ||  PF-2341066 (also see: Crizotinib)  (tyrosine kinase inhibitor)

202223  ||  PF-299804 (not available)

202225  ||  PF-337210

202221  ||  PF-4217903 ( MET tyrosine kinase inhibitor)

202227  ||  PF-477736

202651  ||  PF-4929113 (also see: SNX-5422)

202228  ||  PF-562271 (also see: PF-00562271)

200750  ||  PG-11047 (also see: CGC-11047)

202231  ||  PHA-665752

202233  ||  PHA-848125

202180  ||  Phenoxodiol

202242  ||  Photochlor

202234  ||  PHY-906

202235  ||  PI-103

202230  ||  Picoplatin

202238  ||  PIK-75 (PI3K inhibitor)

202240  ||  Pipendoxifene

202250  ||  Pixantrone

201850  ||  PKC412(also see: Midostaurin )

202255  ||  PKI-587 (also see: PF-05212384)

202260  ||  Plerixafor

202270  ||  Plevitrexed (also see: BGC-9331)

202040  ||  Plinabulin (also see: NPI-2358)

200150  ||  Plitidepsin (also see: Aplidine)

205592  ||  PLX-3397

205611  ||  PLX3603 (also see: RG-7256, RO5212054)

202271  ||  PLX4032 (also see: RG7204, VemurafenibRO5185426)  (B-Raf inhibitor)

202272  ||  PLX-4720 (B-Raf inhibitor)

202290  ||  PM-00104

205594  ||  PM-01183

202300  ||  PM-02734 (also see: Elisidepsin)

205595  ||  PM-060184

202301  ||  PN-401

205596  ||  PNT-2258 (an oligonucleotide therapeutic encapsulated within a SMARTICLES formulation).

205514  ||  PNU-93914 (liposomal paclitaxel, also see: LEP-ETU)

202302  ||  Polyphenon E

202310  ||  Pomalidomide

202320  ||  Ponatinib (also see: AP-24534) (tyrosine kinase inhibitor)

202324  ||  PP242 (mTOR inhibitor)

202330  ||  PPI-2458

202331  ||  PR-104

205626  ||  Pracinostat (also see: SB939)

202320  ||  Pralatrexate

202332  ||  Prinomastat

202334  ||  PRLX-93936

205597  ||  PRT-062607

205598  ||  PRX-302 (protein drug)

202572  ||  PS-095760 (also see: SCH-727965, Dinaciclib) (CDK inhibitor)

205599  ||  PTC-299 (VEGF inhibitor)

205601  ||  PTI-188 (a radiolabeled murine anti-melanin antibody)

205602  ||  PV-10

202340  ||  PX-12

202350  ||  PX-478 (HIF-1alpha inhibitor)

202360  ||  PX-866

202370  ||  Pyroxamide

205603  ||  QBI-139 (protein drug)

201724  ||  QLT-0074 (also see: Lemuteporfin)

202380  ||  Quarfloxin (also see: CX-3543)

202385  ||  Quinacrine(also see: Mepacrine ; CBLC102)

202390  ||  Quinagolide hydrochloride

200072  ||  Quizartinib (also see: AC220) (FLT3 inhibitor)

202391  ||  R1530 (Mitosis-angiogenesis inhibitor)

201650  ||  R1645 (also see: KOS-1584)

200284  ||  R1668 (also see:  ARQ-501,  beta-lapachone)

202411  ||  R306465

202412  ||  R4733 (also see: RO4929097)

202420  ||  R547

202421  ||  R7112 (also see:  RG7112, RO5045337)

202422  ||  R763 (also see: AS703569)

200770  ||  RAF-265 (also  see: CHIR-265)

202430  ||  RC3095

202431  ||  RDEA119 (also see: BAY86-9766) (MEK inhibitor)

202432  ||  RDEA-436

202436  ||  Regorafenib (also see: BAY 73-4506) (oral multi-kinase inhibitor)

202440  ||  Relacatib

202701  ||  Resveratrol(also see: RM1812 , SRT-501)

202450  ||  Retaspimycin (also see: IPI504) (HSP90 inhibitor)

203500  ||  RG3616 (also see: Vismodegib , GDC-0449) (Hedgehog antagonist)

202421  ||  RG7112(also see:  R7112 , RO5045337)

205609  ||  RG-7167

202271  ||  RG7204 (also see: PLX4032, Vemurafenib, RO5185426) (B-Raf inhibitor)

205611  ||  RG-7256 (also see: PLX3603, RO5212054)

205612  ||  RG7304 (also see: CKI27)

205613  ||  RG-7347 (MNRP1685, R7347, Anti-NRP1)

205470  ||  RG7422 (also see: GDC-0980)  (PI3 kinase/mTOR inhibitor)

205615  ||  RG7593 (anti-CD22-MCC-MMAE)

205616  ||  RG7594 (antibody drug)

205240  ||  RG7686 (also see: ECC-33) [monoclonal antibody]

202460  ||  RH1

200860  ||  Ridaforolimus (also see: Deforolimus)

202080  ||  Rigosertibalso see: ON-01910 )

205617  ||  Rindopepimut  (immunotherapy, vaccine)

202701  ||  RM1812 (also see: resveratrol, SRT-501)

202412  ||  RO4929097 (also see: R4733)

202462  ||  RO4987655

202421  ||  RO5045337 (also see:  RG7112, R7112)

202271  ||  RO5185426 (also see: RG7204, Vemurafenib, PLX4032) (B-Raf inhibitor)

205611  ||  RO5212054 (also see: PLX3603, RG-7256)

202470  ||  Rolapitant

202490  ||  Ropidoxuridine

202500  ||  Roquinimex

202510  ||  Rosabulin

202514  ||  Rostaporfin

202520  ||  RP-101 (also see:  Brivudin)

202530  ||  RTA402 (also see: Bardoxolone methyl)

202540  ||  Rubitecan

200124  ||  Rucaparib (Also see: PF-01367338, AG-14699) (PARP1 inhibitor)

201512  ||  Ruxolitinib (also see: INCB-18424) (JAK1 inhibitor)

205618  ||  RX-0201 (Akt antisense oligonucleotide)

202541  ||  S31-201

203210  ||  Sagopilone (also see: ZK epothilone)

202551  ||  Salirasib

202560  ||  Sapacitabine

205619  ||  SAR103168

203181  ||  SAR-245408 (also see: XL147) (PI3K inhibitor)

203187  ||  SAR-245409 (also see: XL765)  (PI3K/mTOR inhibitor)

205620  ||  SAR256212 (also see: MM-121, human monoclonal antibody)

205622  ||  SAR307746 (also see: REGN901, anti-ANG2 monoclonal antibody)

205623  ||  SAR3419

205624  ||  SAR411298 (FAAH inhibitor. Cancer pain)

200410  ||  Saracatinib (also see: AZD-0530) (Src and Abl inhibitor)

200411  ||  Sardomozide

202570  ||  Satraplatin

202571  ||  SB1518 (also see: Pacritinib)

205625  ||  SB1578 (also see: ONX 0805)

205626  ||  SB939 (also see: Pracinostat)

202572  ||  SCH-727965 (also see: Dinaciclib, PS-095760) (CDK inhibitor)

202573  ||  SCH900776 (Chk1 inhibitor)

205572  ||  SDM-230 (also see: Pasireotide)

202580  ||  Seliciclib

200300  ||  Selumetinib (also see: AZD-6244) (MEK 1/2 inhibitor)

202590  ||  Semapimod

202600  ||  Seocalcitol (also see: CB1089)

201614  ||  Serdemetan (also see: JNJ-26854165)

205627  ||  SF1 (also see:  Sonoflora 1)

202601  ||  SF1126

200540  ||  SG2000 (also see: BN2629, SJG-136)

205629  ||  SGI-110

205710  ||  SGI-1776 (pan-Pim protein kinase inhibitor)

205630  ||  SGN-75 (anti-CD70 monoclonal antibody)

205715  ||  SGX-523 (Met Inhibitor)

200274  ||  Silatecan (also see: AR-67, also see: DB-67)

202610  ||  Silibinin

202620  ||  Simotaxel

200020  ||  Sivifene

200540  ||  SJG-136 (also see: BN2629, SG2000)

201372  ||  SK1363089 (also see: XL888, Foretinib, GSK089, EXEL-2880) (MET/VEGFR2 inhibitor)

205631  ||  SL-401 (human IL3 recombinantly conjugated to diphtheria toxin).

202630  ||  SN-2310

201266  ||  SNDX-275(also see: MS-275, Entinostat ) (HDAC inhibitor)

202640  ||  SNS-032 (also see: BMS-387032)

202641  ||  SNS-314

202650  ||  SNS-595 (also see: Voreloxin, Vosaroxin)

202651  ||  SNX-5422 (also see: PF-4929113)

202660  ||  Soblidotin

205627  ||  Sonoflora 1 (also see:  SF1)

205632  ||  Sotatercept (also see: ACE-011, human fusion protein )

202110  ||  SPI-153 (also  see: Ozarelix)

202680  ||  SPI-1620

202690  ||  Squalamine

205672  ||  SR13668 (Akt inhibitor)

202700  ||  SR-31747

202701  ||  SRT-501 (also see: resveratrol, RM1812)

202702  ||  SSR97225

202715  ||  STA-1474

202703  ||  STA-9090 (also see: Ganetespib)

202708  ||  Stannsoporfin

200550  ||  STX64 (also see: Irosustat, BN83495)

202710  ||  SU14813

205633  ||  Sufentanil (also see: ARX-02)

202713  ||  Sulforaphane

205634  ||  SYM-004 (anti-EGFR monoclonal antibody mixture)

200720  ||  TAC-101 (also see: Amsilarotene)

202045  ||  TAE684 (also see: NVP-TAE684) (ALK Inhibitor)

202721  ||  TAK-285

205635  ||  TAK-441

205636  ||  TAK-448

202722  ||  TAK-593

202723  ||  TAK-683

200724  ||  TAK-700 (also see: Orteronel )

205637  ||  TAK-701 (anti-HGF monoclonal antibody)

205638  ||  TAK-733

202725  ||  TAK-901

205639  ||  TAK-960

202730  ||  Talabostat

202740  ||  Talampanel

202750  ||  Talaporfin sodium

202770  ||  Talotrexin Ammonium

202760  ||  Taltobulin

202780  ||  Tamibarotene

202790  ||  Tandutinib (also see: MLN0518) (tyrosine kinase inhibitor)

202950  ||  Tanespimycin (also see:  Telatinib) (Hsp90 inhibitor)

202953  ||  Tanomastat (matrix metalloprotease inhibitor)

100803  ||  Tapentadol

202810  ||  Tarenflurbil

202820  ||  Tariquidar (p-glycoprotein inhibitor)

205641  ||  TAS-102

202834  ||  TAS-103 (also see: BMS-247615)

202840  ||  TAS-108

202841  ||  TAS-109

202850  ||  Tasidotin hydrochloride

202851  ||  Tasisulam (also see: LY573636)

202854  ||  Tasocitinib

202852  ||  Tasquinimod (also see: ABR-215050) (angiogenic inhibitor)

202860  ||  Teglarinad chloride (also see: GMX-1777)

202950  ||  Telatinib (also see:  Tanespimycin) (Hsp90 inhibitor)

202865  ||  Temoporfin

202870  ||  Temsirolimus

202880  ||  Terameprocol (transcriptional inhibitor)

202881  ||  Tesetaxel (also see: DJ-927)

202890  ||  Tesmilifene

202900  ||  Tetrandrine

205642  ||  TG-02

202892  ||  TG100-115 (PI3K inhibitor)

202893  ||  TG101348 ( JAK2 inhibitor)

202895  ||  TGX-221 (PI3K inhibitor)

202901  ||  TH-302

205643  ||  TH-9402

205644  ||  Thiarabine

202902  ||  Thymalfasin

201955  ||  Thymectacin (also see: NB-1011).

202921  ||  Tigapotide

202926  ||  Timcodar (also see: VX-853)

202930  ||  Tipifarnib

202940  ||  Tirapazamine (hypoxia toic agent)

200283  ||  Tivantinib (also see: ARQ-197)  (c-Met inhibitor)

202955  ||  Tivozanib (also see: AV-951) (VEGFR inhibitor)

200760  ||  TKI-258 (also see: Dovitinib, CHIR258)

202960  ||  TL-310 (a taxane)

205645  ||  TL-32711

202962  ||  TLC-388

205646  ||  TOK-001 (also see: Galeterone)

202185  ||  Tookad (also see: Padoporfin)

100880  ||  Toremifene

205648  ||  Tosedostat

202963  ||  Totrombopag

201900  ||  Tozasertib (also  see MK-0457;  VX-680)  (Aurora inhibitor)

202964  ||  TPI-287 (also see: ARC-100)

202970  ||  Trabectedin

201458  ||  Trametinib (aslo see: GSK-1120212, JTP-74057) (MEK 1/2 inhibitor)

205649  ||  TRC093 (a humanized IgG1 monoclonal antibody)

205650  ||  TRC102 (also see: Methoxyamine)

205651  ||  TRC105 (human chimeric monoclonal antibody )

205652  ||  Treosulfan

202980  ||  Tretazicar

203000  ||  Triapine

203010  ||  Triciribine (also see: VQD-002) (Akt inhibitor)

203020  ||  Trilostane

203030  ||  Troxacitabine

205654  ||  TRX-518 (ully humanized IgG1 anti-huGITR Mab)

203031  ||  TST-88 (also  see TST-10088, a recombinant protein prodrug based on a plant-derived toxin called ricin)

203040  ||  TSU-68

203055  ||  Tubacin (HDAC6 inhibitor)

205090  ||  TV-1001 (also see: Custiren, also see: OCX-011) [a mixed-backbone antisense oligodeoxynucleotide with chemosensitizing properties.]

205655  ||  TXA127

205656  ||  U3-1565 (anti-HBEGF monoclonal antibody)

203060  ||  UCN-01(also  see KRX-0601)

203070  ||  Ukrain

203071  ||  UNBS-5162

203080  ||  Uracil

203090  ||  Uridine triacetate

203091  ||  Ursodeoxycholic acid ( also see: Ursodiol)

203091  ||  Ursodiol ( also see: Ursodeoxycholic acid)

205658  ||  V503 (human papillomavirus vaccine)

205659  ||  V935 (hTERT vaccine)

201050  ||  Vadimezan (also see: DMXAA)

203104  ||  Valspodar

203100  ||  Vandetanib (approved in 2011) (VEGFR and EGFR inhibitor)

205660  ||  Varlitinib ( also see: ARRY-543)

203110  ||  Vatalanib (VEGFR inhibitor)

203111  ||  VEL-0230 (also see: NC-2300)

203115  ||  Veliparib (also see:  ABT-888) (PARP inhibitor)

202271  ||  Vemurafenib (also see: RG7204, PLX4032, RO5185426) (B-Raf inhibitor)

200371  ||  VER-52296 (also see: NVP-AUY922,  AUY-922) (Hsp90 inhibitor)

203120  ||  Verteporfin (PDT photosensitizer)

201960  ||  Verubulin (also see: MPC-6827)

203130  ||  Vestipitant

203150  ||  Vinflunine

205661  ||  Virulizin (A natural biological response modifier (BRM) isolated from bovine reticuloendothelial tissue).

203500  ||  Vismodegib (also see: RG3616, GDC-0449)  (Hedgehog antagonist)

200494  ||  Volasertib (also see: BI-6727) (Plk1 inhibitor)

202650  ||  Voreloxin (also see: SNS-595, Vosaroxin)

202650  ||  Vosaroxin (also see: Voreloxin, SNS-595)

203152  ||  VP-701 (not available)

203010  ||  VQD-002 (also see: Triciribine ) (Akt inhibitor)

203153  ||  VTX-2337

201900  ||  VX-680 (also  see MK-0457;  Tozasertib) (Aurora inhibitor)

201917  ||  VX-689 (also see: MK-5108)

203162  ||  VX-702 (p38 MAPK Inhibitor)

203163  ||  VX-745

203165  ||  VX-765 (Caspase inhibitor)

202926  ||  VX-853 (also see: Timcodar)

200390  ||  VX-944 (also see: AVN-944) (IMPDH inhibitor)

203160  ||  WX-671 (also see: Mesupron)

203170  ||  WZ4002 (EGFR inhibitor)

205663  ||  X-82

203180  ||  Xaliproden

205664  ||  Xen-2174 (conopeptide analog)

200535  ||  XL-139 (also see: BMS-833923)

203181  ||  XL147 (also see: SAR-245408) (PI3K inhibitor)

200595  ||  XL-184 (also see:  Cabozantinib)  (VEGFR2, Met, FLT3, Tie2, Kit and Ret inhibitor)

203183  ||  XL228

204730  ||  XL281 (also see:   BMS-908662)

203185  ||  XL518 (also see: GDC-0973)

203186  ||  XL647 (EGFR and ErbB2 inhibitor)

203187  ||  XL765 (also see: SAR-245409) (PI3K/mTOR inhibitor)

201372  ||  XL888 (also see: Foretinib, SK1363089, GSK089, EXEL-2880) (MET/VEGFR2 inhibitor)

205665  ||  XL999

203188  ||  XMT-1001

205666  ||  XMT-1107

200585  ||  XRP-6258 (also see: Cabazitaxel)

201710  ||  XRP9881(also see: Larotaxel )

203190  ||  YM-155 (Survivin inhibitor)

203200  ||  ZD4054 (also see: Zibotentan,  AZD-4054)

200115  ||  ZEN012 (also see: AEZS-112)

203200  ||  Zibotentan (also see: AZD-4054,  ZD4054)

200850  ||  ZIO-101(also see: Darinaparsin )

202130  ||  ZIO-201 (also see: Palifosfamide)

201530  ||  ZIO-301 (also see:Indibulin)

203210  ||  ZK epothilone (also see: Sagopilone)

203215  ||  ZM447439

203220  ||  Zosuquidar trihydrochloride

205668  ||  ZYC-300 (A plasmid DNA)

 

 

 

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