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Approved anticancer agents

Anticancer agents in trials

Anticancer agents in preclinical trials

Anticancer molecular libraries

 


Other drug agents

Drug intermediates

Bio-reagents and biochemicals

 


 

 

 

 

 

MedKoo's

Anticancer molecular libraries

  

EGFR (HER) inhibitors

 

AEE788 (EGFR, ErbB2, KDR, and Flt-1 inhibitor)

Afatinib (EGFR/HER2 inhibitor)

AG-1478 (EGFR inhibitor)

AG-490 (EGFR and JAK inhibitor)

AV-412  (EGFR/HER2 tyrosine kinase inhibitor)

AZD-8931  (HER1and HER2 inhibitor)

BMS-599626 (AC480) (HER1and HER2 inhibitor)

Chrysophanic acid (Chrysophanol ) (EGFR/mTOR pathway inhibitor)

CUDC-101  (HDAC, EGFR and HER2 inhibitor)

Dacomitinib (also see: PF-00299804) (EGFR inhibitor)

Erlotinib (HER1/EGFR TK inhibitor)

Gefitinib  (EGFR inhibitor)

Lapatinib  (EGFR and HER2 inhibitor)

MP-412  (EGFR/HER2 tyrosine kinase inhibitor)

Mubritinib (TAK-165) (EGFR inhibitor)

Neratinib  (HKI272) (HER2 and EGFR inhibitor)

OSI-420 (CP-473420) ( EGFR inhibitor )

PD-153035 (EGFR inhibitor)  

Pelitinib (EKB569) (pan-ErbB tyrosine kinase inhibitor)

PP121(multitargeted dual receptor tyrosine kinases inhibitor )

Vandetanib  (VEGFR and EGFR inhibitor)

WZ3146 (EGFR inhibitor)

WZ4002 (EGFR inhibitor)

WZ8040 ( EGFR inhibitor)

XL647 (EGFR and ErbB2 inhibitor)

  

 

 

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